Development of Poly (ADP-Ribose)Polymerase (PARP) Inhibitors in Oncology

被引:3
作者
Jones, Philip [1 ]
机构
[1] Merck Res Labs Boston, Boston, MA 02115 USA
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 45 | 2010年 / 45卷
关键词
POLY(ADP-RIBOSE) POLYMERASE PARP; POTENT INHIBITORS; DNA-DAMAGE; MAMMARY-TUMORS; MUTANT-CELLS; COMBINATION; DISCOVERY; SENSITIVITY; ABT-888; PHTHALAZINONES;
D O I
10.1016/S0065-7743(10)45014-9
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:229 / +
页数:16
相关论文
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