Solid-phase synthesis of isoxazole-based amino acids: A new scaffold for molecular diversity

被引:25
|
作者
De Luca, L [1 ]
Giacomelli, G [1 ]
Riu, A [1 ]
机构
[1] Univ Sassari, Dipartimento Chim, I-07100 Sassari, Italy
来源
JOURNAL OF ORGANIC CHEMISTRY | 2001年 / 66卷 / 20期
关键词
D O I
10.1021/jo015758v
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:6823 / 6825
页数:3
相关论文
共 50 条
  • [1] Molecular diversity and solid-phase synthesis
    Bondy, S
    Cheng, S
    Saunders, J
    Tarby, C
    Wheeler, K
    DRUG DISCOVERY TODAY, 1996, 1 (04) : 132 - 133
  • [2] N-Fmoc-dehydroalanine:: a versatile molecular scaffold for the rapid solid-phase synthesis of cycloaliphatic amino acids
    Burkett, BA
    Chai, CLL
    TETRAHEDRON LETTERS, 2000, 41 (34) : 6661 - 6664
  • [3] Solid-phase synthesis of α,α-difluorinated β-amino acids by Reformatsky reaction
    Nefzi, A
    Vidal, A
    Houghten, RA
    BIOPOLYMERS, 2003, 71 (03) : 353 - 353
  • [4] Amino monothio acids in solid-phase synthesis of peptide thioamides
    HoegJensen, T
    Spatola, AF
    Holm, A
    INTERNATIONAL JOURNAL OF PEPTIDE AND PROTEIN RESEARCH, 1996, 47 (03): : 190 - 200
  • [5] Solid-phase synthesis of liquid crystalline isoxazole library
    Haino, T
    Tanaka, M
    Ideta, K
    Kubo, K
    Mori, A
    Fukazawa, Y
    TETRAHEDRON LETTERS, 2004, 45 (11) : 2277 - 2279
  • [6] Molecular Diversity of Hydroxamic Acids: Part I. Solution- and Solid-Phase Synthesis
    Yang, Kexin
    Lou, Boliang
    MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2003, 3 (04) : 349 - 360
  • [7] Molecular diversity of peptidomimetics: Approaches to the solid-phase synthesis of peptidosulfonamides
    deBont, DBA
    Moree, WJ
    Liskamp, RMJ
    BIOORGANIC & MEDICINAL CHEMISTRY, 1996, 4 (05) : 667 - 672
  • [8] Synthesis, biological evaluation, molecular docking, and ADMET studies of some isoxazole-based amides
    Sushama Kauthale
    Sunil Tekale
    Manoj Damale
    Jaiprakash Sangshetti
    Rajendra Pawar
    Medicinal Chemistry Research, 2018, 27 : 429 - 441
  • [9] Solid-phase peptide synthesis using nanoparticulate amino acids in water
    Hojo, Keiko
    Ichikawa, Hideki
    Iviaeda, Mitsuko
    Kida, Shinya
    Fukumori, Yoshinobu
    Kawasaki, Koichi
    JOURNAL OF PEPTIDE SCIENCE, 2007, 13 (07) : 493 - 497
  • [10] Solid-phase synthesis of α-amino acids by radical addition to a dehydroalanine derivative
    Yim, AM
    Vidal, Y
    Viallefont, P
    Martinez, J
    TETRAHEDRON LETTERS, 1999, 40 (24) : 4535 - 4538