3-Bromocyclohexane-1,2-dione as a useful reagent for Hantzsch synthesis of thiazoles and the synthesis of related heterocycles

被引：17
作者：
Guernon, Jason M. [1 ]
Wu, Yong-Jin [1 ]
机构：
[1] Bristol Myers Squibb Co, Dept Neurosci Chem, Res & Dev, Wallingford, CT 06492 USA
来源：
TETRAHEDRON LETTERS | 2011年 / 52卷 / 28期
关键词：
3-Bromocyclohexan-1,2-dione; Hantzsch; Thiazole; SERIES;
D O I：
10.1016/j.tetlet.2011.05.028
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
We describe the use of 3-bromocyclohexane-1,2-dione, an air stable, versatile reagent for the Hantzsch thiazole synthesis and the synthesis of other closely related heterocycles. (C) 2011 Elsevier Ltd. All rights reserved.
引用
收藏
页码：3633 / 3635
页数：3
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