When and How to Use Somatostatin Analogues

被引：10
作者：
de Herder, Wouter W. [1 ]
机构：
[1] Erasmus MC, Dept Internal Med, Sect Endocrinol, ENETS Ctr Excellence Neuroendocrine Tumors, Dr Molewaterpl 40, NL-3015 GD Rotterdam, Netherlands
来源：
ENDOCRINOLOGY AND METABOLISM CLINICS OF NORTH AMERICA | 2018年 / 47卷 / 03期
关键词：
Somatostatin; Receptor; Octreotide; Lanreotide; Pasireotide; Neuroendocrine; GASTROENTEROPANCREATIC NEUROENDOCRINE TUMORS; RECEPTOR RADIONUCLIDE THERAPY; ENETS CONSENSUS GUIDELINES; LONG-ACTING PASIREOTIDE; CUSHINGS-SYNDROME; CARCINOID-SYNDROME; GASTROINTESTINAL-TRACT; OCTREOTIDE LAR; MANAGEMENT; EVEROLIMUS;
D O I：
10.1016/j.ecl.2018.04.010
中图分类号：
R5 [内科学];
学科分类号：
1002 ; 100201 ;
摘要：
Long-acting depot formulations of the currently available somatostatin analogues are considered the first-line treatment for control of hormonal excess by hormone-producing neuroendocrine tumors of the gastrointestinal tract and pancreas. These drugs are currently also considered the first-line treatment for tumor control of both hormone-producing and non-hormone-producing neuroendocrine tumors of the gastrointestinal tract and pancreas. These drugs need coupling and interaction with specific somatostatin receptor subtypes, which are expressed on the cells of neuroendocrine tumors of the gastrointestinal tract and pancreas.
引用
收藏
页码：549 / +
页数：8
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