Synthesis and antibacterial activity of 2-(3-acylphenyl)amino-4-phenylthiazole

被引：0

作者：

Subhashini, N. J. P. ^{[1
]}

Amanaganti, Jampaiah ^{[1
]}

Shivaraj ^{[1
]}

机构：

[1] Osmania Univ, Dept Chem, Univ Coll Technol, Hyderabad 500007, Andhra Pradesh, India

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2015年 / 85卷 / 03期

关键词：

thiazoles; 1-(3-acetylphenyl)thiourea; 2-bromo-1-phenylethanone; antibacterial activity; DERIVATIVES;

D O I：

10.1134/S1070363215030275

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

2-(3-acylphenyl)amino-4-phenylthiazoles were synthesized from 1-(3-acetylphenyl)thiourea and 2-bromo-1-substituted phenylethanones in presence of triethylamine upon heating. The newly synthesized compounds were characterized by IR, H-1 NMR, MS spectrometry. All products were evaluated for their antibacterial activity against Gram positive (Staphylococcus aureus and Bacillus subtilis) and Gram negative (Escherichia coli, Klebsiella pnemoniae) strains.

引用

页码：686 / 688

页数：3

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