3-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]-1H-pyrrolo[2,3-b]pyridine: An antagonist with high affinity and selectivity for the human dopamine D-4 receptor

被引:253
作者
Kulagowski, JJ
Broughton, HB
Curtis, NR
Mawer, IM
Ridgill, MP
Baker, R
Emms, F
Freedman, SB
Marwood, R
Patel, S
Patel, S
Ragan, CI
Leeson, PD
机构
[1] Merck Sharp and Dohme Res. Labs., Neuroscience Research Centre, Harlow, Essex CM20 2QR, Terlings Park, Eastwick Road
关键词
D O I
10.1021/jm9600712
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:1941 / 1942
页数:2
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