Covalently induced activation of the δ opioid receptor by a fluorogenic affinity label, 7′-(phthalaldehyde-carboxamido)naltrindole (PNTI)

被引：10

作者：

Le Bourdonnec, B

El Kouhen, R

Poda, G

Law, PY

Loh, HH

Ferguson, DM

Portoghese, PS ^{[1
]}

机构：

[1] Univ Minnesota, Coll Pharm, Dept Med Chem, Minneapolis, MN 55455 USA

[2] Univ Minnesota, Sch Med, Dept Pharmacol, Minneapolis, MN 55455 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2001年 / 44卷 / 07期

关键词：

D O I：

10.1021/jm010004u

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1017 / 1020

页数：4

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