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- [1] A first-in-human phase I study to evaluate GDC-0980, an oral PI3K/mTOR inhibitor, administered QD in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2011, 29 (15)Wagner, A. J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USABendell, J. C.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USADolly, S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAMorgan, J. A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAWare, J. A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAFredrickson, J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAMazina, K. E.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USALauchle, J. O.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USABurris, H. A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USADe Bono, J. S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA
- [2] A phase I study evaluating the pharmacokinetics (PK) and pharmacodynamic (PD) activity of the dual PI3K/mTor inhibitor GDC-0980 administered QWEJC SUPPLEMENTS, 2010, 8 (07): : 123 - 124Wagner, A. J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAJayson, G. C.论文数: 0 引用数: 0 h-index: 0机构: Christie NHS Fdn Trust, Manchester, Lancs, England Dana Farber Canc Inst, Boston, MA 02115 USAGomez-Roca, C.论文数: 0 引用数: 0 h-index: 0机构: Inst Cancerol Gustave Roussy, Villejuif, France Dana Farber Canc Inst, Boston, MA 02115 USAZee, Y. K.论文数: 0 引用数: 0 h-index: 0机构: Christie NHS Fdn Trust, Manchester, Lancs, England Dana Farber Canc Inst, Boston, MA 02115 USAMorgan, J. A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAYan, Y.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, GRED, San Francisco, CA 94080 USA Dana Farber Canc Inst, Boston, MA 02115 USAWare, J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, GRED, San Francisco, CA 94080 USA Dana Farber Canc Inst, Boston, MA 02115 USAMazina, K. E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, GRED, San Francisco, CA 94080 USA Dana Farber Canc Inst, Boston, MA 02115 USALauchle, J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, GRED, San Francisco, CA 94080 USA Dana Farber Canc Inst, Boston, MA 02115 USASoria, J. C.论文数: 0 引用数: 0 h-index: 0机构: Inst Cancerol Gustave Roussy, Villejuif, France Dana Farber Canc Inst, Boston, MA 02115 USA
- [3] Discovery of GDC-0980, a selective PI3K/mTOR inhibitor in clinical trialsCANCER RESEARCH, 2011, 71Sutherlin, Daniel P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABelvin, Marcia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABao, Linda论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABerry, Leanne论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABerry, Megan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USACastanedo, Georgette论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAEdgar, Kyle论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAFolkes, Adrian论文数: 0 引用数: 0 h-index: 0机构: Plramed, Slough, Berks, England Genentech Inc, San Francisco, CA 94080 USAFriedman, Lori论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHeffron, Tim论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAPatel, Sonal论文数: 0 引用数: 0 h-index: 0机构: Plramed, Slough, Berks, England Genentech Inc, San Francisco, CA 94080 USAOlivero, Alan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALesnick, John论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALewis, Cristina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAMarsters, James论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USANonomiya, Jim论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAPang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAPrior, Wei Wei论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASampath, Deepak论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USATsui, Vickie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWallin, Jeff论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWei, BinQing论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWeismann, Christian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAZhu, Bing-Yan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [4] Process development of PI3K inhibitor GDC-0980ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Humphries, Theresa论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Proc Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Proc Chem, San Francisco, CA 94080 USA
- [5] A novel potent and selective inhibitor of PI3K/mTOR, GDC-0980, currently in phase I clinical trialsMOLECULAR CANCER THERAPEUTICS, 2009, 8 (12)Friedman, Lori S.论文数: 0 引用数: 0 h-index: 0Belvin, Marcia论文数: 0 引用数: 0 h-index: 0Berry, Leanne论文数: 0 引用数: 0 h-index: 0Berry, Megan论文数: 0 引用数: 0 h-index: 0Castanedo, Georgette论文数: 0 引用数: 0 h-index: 0Edgar, Kyle论文数: 0 引用数: 0 h-index: 0Folkes, Adrian论文数: 0 引用数: 0 h-index: 0Guan, Jane论文数: 0 引用数: 0 h-index: 0Heffron, Tim论文数: 0 引用数: 0 h-index: 0Lesnick, John论文数: 0 引用数: 0 h-index: 0Lewis, Cris论文数: 0 引用数: 0 h-index: 0Nonomiya, Jim论文数: 0 引用数: 0 h-index: 0Olivero, Alan论文数: 0 引用数: 0 h-index: 0Patel, Sonal论文数: 0 引用数: 0 h-index: 0Pang, Jodie论文数: 0 引用数: 0 h-index: 0Prior, Wei Wei论文数: 0 引用数: 0 h-index: 0Salphati, Laurent论文数: 0 引用数: 0 h-index: 0Sampath, Deepak论文数: 0 引用数: 0 h-index: 0Sutherlin, Dan论文数: 0 引用数: 0 h-index: 0Wallin, Jeff论文数: 0 引用数: 0 h-index: 0Zhu, Bingyan论文数: 0 引用数: 0 h-index: 0
- [6] Phase II trial of GDC-0980 (dual PI3K/mTOR inhibitor) in patients with advanced endometrial carcinoma: Final study results.JOURNAL OF CLINICAL ONCOLOGY, 2014, 32 (15)Makker, Vicky论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USARecio, Fernando O.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAMa, Ling论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAMatutonis, Ursula论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USALauchle, Jennifer O'Hara论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAParmar, Hema论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAGilbert, Houston论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAWang, Yulei论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAKoeppen, Hartmut论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USASpoerke, Jill M.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USALackner, Mark论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAAghajanian, Carol论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA
- [7] A first-in-human, phase I study to evaluate the dual PI3K/mTOR inhibitor GDC-0980 administered QD in patients with advanced solid tumors or non-Hodgkin's lymphomaJOURNAL OF CLINICAL ONCOLOGY, 2010, 28 (15)Dolly, S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandWagner, A. J.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandBendell, J. C.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandYan, Y.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandWare, J. A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandMazina, K. E.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandHolden, S. N.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandDerynck, M. K.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandDe Bono, J. S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, EnglandBurris, H. A., III论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, London SW3 6JJ, England
- [8] POPULATION PHARMACOKINETICS AND PHARMACODYNAMICS OF THE PAN-PHOSPHOINOSITIDE-3 KINASE (PI3K) INHIBITOR GDC-0941 IN PHASE I PATIENTS WITH ADVANCED SOLID TUMORSCLINICAL PHARMACOLOGY & THERAPEUTICS, 2011, 89 : S81 - S81Lin, J. Y.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABudha, N.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWare, J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWest, D.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAIginla, S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAYan, Y.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHolden, S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADerynck, M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADresser, M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADresser, M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [9] A FIRST-IN-HUMAN PHASE I STUDY TO EVALUATE THE DUAL PI3K/MTOR INHIBITOR GDC-0980 ADMINISTERED QD IN PATIENTS WITH ADVANCED SOLID TUMORS OR NON-HODGKIN S LYMPHOMA (NHL)ANNALS OF ONCOLOGY, 2010, 21 : 162 - 163Bendell, J. C.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Sarah Cannon Res Inst, Nashville, TN USAWagner, A. J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Sarah Cannon Res Inst, Nashville, TN USADolly, S.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAMorgan, J. A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Sarah Cannon Res Inst, Nashville, TN USAPapadatos-Pastos, D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Inst Canc Res, Drug Dev Unit, Sutton, Surrey, England Sarah Cannon Res Inst, Nashville, TN USAWare, J.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAMazina, K. E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Res & Early Dev, San Francisco, CA 94080 USA Sarah Cannon Res Inst, Nashville, TN USALauchle, J.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USABurris, H.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Sarah Cannon Res Inst, Nashville, TN USADe Bono, J.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Inst Canc Res, Drug Dev Unit, Sutton, Surrey, England Sarah Cannon Res Inst, Nashville, TN USA
- [10] GDC-0980 Is a Novel Class I PI3K/mTOR Kinase Inhibitor with Robust Activity in Cancer Models Driven by the PI3K PathwayMOLECULAR CANCER THERAPEUTICS, 2011, 10 (12) : 2426 - 2436Wallin, Jeffrey J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAEdgar, Kyle A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAGuan, Jane论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USABerry, Megan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAPrior, Wei Wei论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USALee, Leslie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USALesnick, John D.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Biomed Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USALewis, Cristina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Biomed Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USANonomiya, Jim论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Biomed Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAPang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAOlivero, Alan G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USASutherlin, Daniel P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAO'Brien, Carol论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Dev Oncol Diagnost, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USASpoerke, Jill M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Dev Oncol Diagnost, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAPatel, Sonal论文数: 0 引用数: 0 h-index: 0机构: Piramed, Slough, Berks, England Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USALensun, Letitia论文数: 0 引用数: 0 h-index: 0机构: Piramed, Slough, Berks, England Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAKassees, Robert论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USARoss, Leanne论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USALackner, Mark R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Dev Oncol Diagnost, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USASampath, Deepak论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USABelvin, Marcia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USAFriedman, Lori S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA