Design, antiviral and pharmacokinetic profiles of potent 1,3,4-trisubstituted pyrrolidine CCR5 receptor antagonists for the treatment of HIV-1 infection.
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作者:
Kim, D
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Kim, D
Wang, LP
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Wang, LP
Hale, JJ
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Hale, JJ
Lynch, C
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Lynch, C
Budhu, RJ
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Budhu, RJ
MacCoss, M
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
MacCoss, M
Mills, SG
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Mills, SG
Malkowitz, L
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Malkowitz, L
Gould, SL
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Gould, SL
DeMartino, JA
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
DeMartino, JA
Springer, MS
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Springer, MS
Hazuda, D
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Hazuda, D
Kessler, J
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Kessler, J
Danzeisen, R
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Danzeisen, R
Carella, A
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Carella, A
Holmes, K
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Holmes, K
Lineberger, J
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Lineberger, J
Schleif, WA
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Schleif, WA
Emini, EA
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机构:Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
Emini, EA
机构:
[1] Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
[2] Merck Res Labs, Dept Immunol, Rahway, NJ 07065 USA
[3] Merck Res Labs, Dept Antiviral Res, Rahway, NJ 07065 USA
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