MEDI 93-MDM2 inhibitory peptides: Side chains cyclization as a method of stabilization of the biologically active helical conformation
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作者:
Krajewski, Krzysztof
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NCI, Med Chem Lab, NIH, Frederick, MD 21702 USANCI, Med Chem Lab, NIH, Frederick, MD 21702 USA
Krajewski, Krzysztof
[1
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Nikolovska-Coleska, Zaneta
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Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USANCI, Med Chem Lab, NIH, Frederick, MD 21702 USA
Nikolovska-Coleska, Zaneta
[2
,3
,4
,5
]
Wang, Shaomeng
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Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USANCI, Med Chem Lab, NIH, Frederick, MD 21702 USA
Wang, Shaomeng
[2
,3
,4
,5
]
Roller, Peter P.
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NCI, Med Chem Lab, NIH, Frederick, MD 21702 USANCI, Med Chem Lab, NIH, Frederick, MD 21702 USA
Roller, Peter P.
[1
]
机构:
[1] NCI, Med Chem Lab, NIH, Frederick, MD 21702 USA
[2] Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
[3] Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
[4] Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA
[5] Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA
机构:
Indian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India
Sri Guru Granth Sahib World Univ, Sch Basic & Appl Sci, Dept Chem, Fatehgarh Sahib 140406, Punjab, IndiaIndian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India
Goyal, Bhupesh
Srivastava, Kinshuk Raj
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Indian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India
Univ Michigan, Inst Life Sci, Ann Arbor, MI 48105 USAIndian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India
Srivastava, Kinshuk Raj
Durani, Susheel
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Indian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, IndiaIndian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India