Iron(II) Triflate as a Catalyst for the Synthesis of Indoles by Intramolecular C-H Amination

被引：136
作者：
Bonnamour, Julien [1 ]
Bolm, Carsten [1 ]
机构：
[1] Rhein Westfal TH Aachen, Inst Organ Chem, D-52056 Aachen, Germany
来源：
ORGANIC LETTERS | 2011年 / 13卷 / 08期
关键词：
CROSS-COUPLING REACTIONS; AZIRIDINATION REACTIONS; ORGANIC-SYNTHESIS; METAL-COMPLEXES; ARYL AZIDES; SULFIDES; SULFOXIDES; AZIDOACRYLATES; REARRANGEMENT; 2H-AZIRINES;
D O I：
10.1021/ol2004066
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A practical iron-catalyzed intramolecular C-H amination reaction and its application in the synthesis of indole derivatives are presented. As a catalyst, commercially available iron(II) triflate is used.
引用
收藏
页码：2012 / 2014
页数：3
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