Targeting PI3K/AKT pathway in triple-negative breast cancer

被引:39
作者
Delaloge, Suzette [1 ]
DeForceville, Louise [1 ]
机构
[1] Gustave Roussy, Dept Med Oncol, F-94800 Villejuif, France
关键词
TUMORS;
D O I
10.1016/S1470-2045(17)30514-4
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:1293 / 1294
页数:3
相关论文
共 7 条
[1]   Triple-negative breast cancer: challenges and opportunities of a heterogeneous disease [J].
Bianchini, Giampaolo ;
Balko, Justin M. ;
Mayer, Ingrid A. ;
Sanders, Melinda E. ;
Gianni, Luca .
NATURE REVIEWS CLINICAL ONCOLOGY, 2016, 13 (11) :674-690
[2]   A Randomized Phase II Neoadjuvant Study of Cisplatin, Paclitaxel With or Without Everolimus in Patients with Stage II/III Triple-Negative Breast Cancer (TNBC): Responses and Long-term Outcome Correlated with Increased Frequency of DNA Damage Response Gene Mutations, TNBC Subtype, AR Status, and Ki67 [J].
Jovanovic, Bojana ;
Mayer, Ingrid A. ;
Mayer, Erica L. ;
Abramson, Vandana G. ;
Bardia, Aditya ;
Sanders, Melinda E. ;
Kuba, M. Gabriela ;
Estrada, Monica V. ;
Beeler, J. Scott ;
Shaver, Timothy M. ;
Johnson, Kimberly C. ;
Sanchez, Violeta ;
Rosenbluth, Jennifer M. ;
Dillon, Patrick M. ;
Forero-Torres, Andres ;
Chang, Jenny C. ;
Meszoely, Ingrid M. ;
Grau, Ana M. ;
Lehmann, Brian D. ;
Shyr, Yu ;
Sheng, Quanhu ;
Chen, Sheau-Chiann ;
Arteaga, Carlos L. ;
Pietenpol, Jennifer A. .
CLINICAL CANCER RESEARCH, 2017, 23 (15) :4035-4045
[3]  
Kim SB, 2017, LANCET ONCOL
[4]   Comprehensive molecular portraits of human breast tumours [J].
Koboldt, Daniel C. ;
Fulton, Robert S. ;
McLellan, Michael D. ;
Schmidt, Heather ;
Kalicki-Veizer, Joelle ;
McMichael, Joshua F. ;
Fulton, Lucinda L. ;
Dooling, David J. ;
Ding, Li ;
Mardis, Elaine R. ;
Wilson, Richard K. ;
Ally, Adrian ;
Balasundaram, Miruna ;
Butterfield, Yaron S. N. ;
Carlsen, Rebecca ;
Carter, Candace ;
Chu, Andy ;
Chuah, Eric ;
Chun, Hye-Jung E. ;
Coope, Robin J. N. ;
Dhalla, Noreen ;
Guin, Ranabir ;
Hirst, Carrie ;
Hirst, Martin ;
Holt, Robert A. ;
Lee, Darlene ;
Li, Haiyan I. ;
Mayo, Michael ;
Moore, Richard A. ;
Mungall, Andrew J. ;
Pleasance, Erin ;
Robertson, A. Gordon ;
Schein, Jacqueline E. ;
Shafiei, Arash ;
Sipahimalani, Payal ;
Slobodan, Jared R. ;
Stoll, Dominik ;
Tam, Angela ;
Thiessen, Nina ;
Varhol, Richard J. ;
Wye, Natasja ;
Zeng, Thomas ;
Zhao, Yongjun ;
Birol, Inanc ;
Jones, Steven J. M. ;
Marra, Marco A. ;
Cherniack, Andrew D. ;
Saksena, Gordon ;
Onofrio, Robert C. ;
Pho, Nam H. .
NATURE, 2012, 490 (7418) :61-70
[5]   A randomized adaptive phase II/III study of buparlisib, a pan-class I PI3K inhibitor, combined with paclitaxel for the treatment of HER2-advanced breast cancer (BELLE-4) [J].
Martin, M. ;
Chan, A. ;
Dirix, L. ;
O'Shaughnessy, J. ;
Hegg, R. ;
Manikhas, A. ;
Shtivelband, M. ;
Krivorotko, P. ;
Batista Lopez, N. ;
Campone, M. ;
Ruiz Borrego, M. ;
Khan, Q. J. ;
Beck, J. T. ;
Ramos Vazquez, M. ;
Urban, P. ;
Goteti, S. ;
Di Tomaso, E. ;
Massacesi, C. ;
Delaloge, S. .
ANNALS OF ONCOLOGY, 2017, 28 (02) :313-320
[6]   Olaparib for Metastatic Breast Cancer in Patients with a Germline BRCA Mutation [J].
Robson, Mark ;
Im, Seock-Ah ;
Senkus, Elzbieta ;
Xu, Binghe ;
Domchek, Susan M. ;
Masuda, Norikazu ;
Delaloge, Suzette ;
Li, Wei ;
Tung, Nadine ;
Armstrong, Anne ;
Wu, Wenting ;
Goessl, Carsten ;
Runswick, Sarah ;
Conte, Pierfranco .
NEW ENGLAND JOURNAL OF MEDICINE, 2017, 377 (06) :523-533
[7]   A First-in-Human Phase I Study of the ATP-Competitive AKT Inhibitor Ipatasertib Demonstrates Robust and Safe Targeting of AKT in Patients with Solid Tumors [J].
Saura, Cristina ;
Roda, Desamparados ;
Rosello, Susana ;
Oliveira, Mafalda ;
Macarulla, Teresa ;
Alejandro Perez-Fidalgo, Jose ;
Morales-Barrera, Rafael ;
Manuel Sanchis-Garcia, Juan ;
Musib, Luna ;
Budha, Nageshwar ;
Zhu, Jin ;
Nannini, Michelle ;
Chan, Wai Y. ;
Bohorquez, Sandra M. Sanabria ;
Meng, Raymond D. ;
Lin, Kui ;
Yan, Yibing ;
Patel, Premal ;
Baselga, Jose ;
Tabernero, Josep ;
Cervantes, Andres .
CANCER DISCOVERY, 2017, 7 (01) :102-113