共 5 条
[1]
Spectrum of Mechanisms of Resistance to Crizotinib and Lorlatinib in ROS1 Fusion-Positive Lung Cancer
[J].
Lin, Jessica J.
;
Choudhury, Noura J.
;
Yoda, Satoshi
;
Zhu, Viola W.
;
Johnson, Ted W.
;
Sakhtemani, Ramin
;
Dagogo-Jack, Ibiayi
;
Digumarthy, Subba R.
;
Lee, Charlotte
;
Do, Andrew
;
Peterson, Jennifer
;
Prutisto-Chang, Kylie
;
Malik, Wafa
;
Hubbeling, Harper G.
;
Langenbucher, Adam
;
Schoenfeld, Adam J.
;
Falcon, Christina J.
;
Temel, Jennifer S.
;
Sequist, Lecia, V
;
Yeap, Beow Y.
;
Lennerz, Jochen K.
;
Shaw, Alice T.
;
Lawrence, Michael S.
;
Ou, Sai-Hong Ignatius
;
Hata, Aaron N.
;
Drilon, Alexander
;
Gainor, Justin F.
.
CLINICAL CANCER RESEARCH,
2021, 27 (10)
:2899-2909

Lin, Jessica J.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Choudhury, Noura J.
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Dept Med, 1275 York Ave, New York, NY 10021 USA
Weill Cornell Med Coll, New York, NY USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Yoda, Satoshi
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Zhu, Viola W.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Irvine, Dept Med, Orange, CA 92668 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Johnson, Ted W.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, La Jolla, CA USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Sakhtemani, Ramin
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Dagogo-Jack, Ibiayi
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Digumarthy, Subba R.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp, Dept Radiol, Boston, MA 02114 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Lee, Charlotte
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Do, Andrew
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Peterson, Jennifer
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Prutisto-Chang, Kylie
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Malik, Wafa
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Hubbeling, Harper G.
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Dept Med, 1275 York Ave, New York, NY 10021 USA
Weill Cornell Med Coll, New York, NY USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Langenbucher, Adam
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Schoenfeld, Adam J.
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Dept Med, 1275 York Ave, New York, NY 10021 USA
Weill Cornell Med Coll, New York, NY USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Falcon, Christina J.
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Dept Med, 1275 York Ave, New York, NY 10021 USA
Weill Cornell Med Coll, New York, NY USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Temel, Jennifer S.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Sequist, Lecia, V
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Yeap, Beow Y.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Lennerz, Jochen K.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Shaw, Alice T.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Lawrence, Michael S.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Ou, Sai-Hong Ignatius
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Irvine, Dept Med, Orange, CA 92668 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Hata, Aaron N.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Drilon, Alexander
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Dept Med, 1275 York Ave, New York, NY 10021 USA
Weill Cornell Med Coll, New York, NY USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA

Gainor, Justin F.
论文数: 0 引用数: 0
h-index: 0
机构:
Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
Harvard Med Sch, Boston, MA 02115 USA Massachusetts Gen Hosp Canc Ctr, Dept Med, Boston, MA USA
[2]
ALKG1269A mutation as a potential mechanism of acquired resistance to crizotinib in an ALK-rearranged inflammatory myofibroblastic tumor
[J].
Michels, Sebastian Y. F.
;
Scheel, Andreas H.
;
Wuendisch, Thomas
;
Heuckmann, Johannes M.
;
Menon, Roopika
;
Puesken, Michael
;
Kobe, Carsten
;
Pasternack, Helen
;
Heydt, Carina
;
Scheffler, Matthias
;
Fischer, Rieke
;
Schultheis, Anne M.
;
Merkelbach-Bruse, Sabine
;
Heukamp, Lukas
;
Buettner, Reinhard
;
Woelf, Jurgen
.
NPJ PRECISION ONCOLOGY,
2017, 1

Michels, Sebastian Y. F.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Ctr Integrated Oncol, Dept Internal Med 1, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Scheel, Andreas H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Inst Pathol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Wuendisch, Thomas
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Dusseldorf, Comprehens Canc Ctr Dusseldorf, Dusseldorf, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Heuckmann, Johannes M.
论文数: 0 引用数: 0
h-index: 0
机构:
NEO New Oncol AG, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Menon, Roopika
论文数: 0 引用数: 0
h-index: 0
机构:
NEO New Oncol AG, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Puesken, Michael
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Dept Radiol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Kobe, Carsten
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Dept Nucl Med, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Pasternack, Helen
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Inst Pathol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Heydt, Carina
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Inst Pathol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Scheffler, Matthias
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Ctr Integrated Oncol, Dept Internal Med 1, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Fischer, Rieke
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Ctr Integrated Oncol, Dept Internal Med 1, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Schultheis, Anne M.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Inst Pathol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Merkelbach-Bruse, Sabine
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Inst Pathol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Heukamp, Lukas
论文数: 0 引用数: 0
h-index: 0
机构:
NEO New Oncol AG, Cologne, Germany
Inst Hematopathol, Hamburg, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Buettner, Reinhard
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Inst Pathol, Ctr Integrated Oncol, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany

Woelf, Jurgen
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
Univ Hosp Cologne, Ctr Integrated Oncol, Dept Internal Med 1, Cologne, Germany Univ Hosp Cologne, Lung Canc Grp Cologne, Cologne, Germany
[3]
US Phase I First-in-human Study of Taletrectinib (DS-6051b/AB-106), a ROS1/TRK Inhibitor, in Patients with Advanced Solid Tumors
[J].
Papadopoulos, Kyriakos P.
;
Borazanci, Erkut
;
Shaw, Alice T.
;
Katayama, Ryohei
;
Shimizu, Yuki
;
Zhu, Viola W.
;
Sun, Thomas Yang
;
Wakelee, Heather A.
;
Madison, Russell
;
Schrock, Alexa B.
;
Senaldi, Giorgio
;
Nakao, Naoki
;
Hanzawa, Hiroyuki
;
Tachibana, Masaya
;
Isoyama, Takeshi
;
Nakamaru, Kenji
;
Deng, Chenhui
;
Li, Meijing
;
Fan, Frank
;
Zhao, Qinying
;
Gao, Yanfei
;
Seto, Takashi
;
Janne, Pasi A.
;
Ou, Sai-Hong Ignatius
.
CLINICAL CANCER RESEARCH,
2020, 26 (18)
:4785-4794

Papadopoulos, Kyriakos P.
论文数: 0 引用数: 0
h-index: 0
机构:
South Texas Accelerated Res Therapeut, San Antonio, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Borazanci, Erkut
论文数: 0 引用数: 0
h-index: 0
机构:
HonorHlth & Translat Genom Res Inst, Scottsdale, AZ USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Shaw, Alice T.
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst BioMed Res, Cambridge, MA USA
Harvard Med Sch, Massachusetts Gen Hosp, Boston, MA 02115 USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Katayama, Ryohei
论文数: 0 引用数: 0
h-index: 0
机构:
Japanese Fdn Canc Res, Ctr Canc Chemotherapy, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Shimizu, Yuki
论文数: 0 引用数: 0
h-index: 0
机构:
Japanese Fdn Canc Res, Ctr Canc Chemotherapy, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Zhu, Viola W.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Irvine, Sch Med, Chao Family Comprehens Canc Ctr, Orange, CA 92868 USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

论文数: 引用数:
h-index:
机构:

Wakelee, Heather A.
论文数: 0 引用数: 0
h-index: 0
机构:
Stanford Univ, Dept Med, Div Oncol, Stanford Canc Inst, Stanford, CA 94305 USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Madison, Russell
论文数: 0 引用数: 0
h-index: 0
机构:
Fdn Med Inc, Cambridge, MA USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Schrock, Alexa B.
论文数: 0 引用数: 0
h-index: 0
机构:
Fdn Med Inc, Cambridge, MA USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Senaldi, Giorgio
论文数: 0 引用数: 0
h-index: 0
机构:
Daiichi Sankyo Inc, Basking Ridge, NJ USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Nakao, Naoki
论文数: 0 引用数: 0
h-index: 0
机构:
Daiichi Sankyo RD Novare Co Ltd, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Hanzawa, Hiroyuki
论文数: 0 引用数: 0
h-index: 0
机构:
Daiichi Sankyo RD Novare Co Ltd, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Tachibana, Masaya
论文数: 0 引用数: 0
h-index: 0
机构:
Daiichi Sankyo Co Ltd, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Isoyama, Takeshi
论文数: 0 引用数: 0
h-index: 0
机构:
Daiichi Sankyo Co Ltd, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Nakamaru, Kenji
论文数: 0 引用数: 0
h-index: 0
机构:
Daiichi Sankyo Co Ltd, Tokyo, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Deng, Chenhui
论文数: 0 引用数: 0
h-index: 0
机构:
Linking Truth Technol Co Ltd, Beijing, Peoples R China South Texas Accelerated Res Therapeut, San Antonio, TX USA

Li, Meijing
论文数: 0 引用数: 0
h-index: 0
机构:
AnHeart Therapeut Hangzhou Co Ltd, Hangzhou, Zhejiang, Peoples R China South Texas Accelerated Res Therapeut, San Antonio, TX USA

Fan, Frank
论文数: 0 引用数: 0
h-index: 0
机构:
AnHeart Therapeut Hangzhou Co Ltd, Hangzhou, Zhejiang, Peoples R China South Texas Accelerated Res Therapeut, San Antonio, TX USA

Zhao, Qinying
论文数: 0 引用数: 0
h-index: 0
机构:
AnHeart Therapeut Hangzhou Co Ltd, Hangzhou, Zhejiang, Peoples R China South Texas Accelerated Res Therapeut, San Antonio, TX USA

Gao, Yanfei
论文数: 0 引用数: 0
h-index: 0
机构:
AnHeart Therapeut Hangzhou Co Ltd, Hangzhou, Zhejiang, Peoples R China South Texas Accelerated Res Therapeut, San Antonio, TX USA

Seto, Takashi
论文数: 0 引用数: 0
h-index: 0
机构:
Natl Hosp Org Kyushu Canc Ctr, Dept Thorac Oncol, Fukuoka, Japan South Texas Accelerated Res Therapeut, San Antonio, TX USA

Janne, Pasi A.
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Med Sch, Dana Farber Canc Inst, Boston, MA 02115 USA South Texas Accelerated Res Therapeut, San Antonio, TX USA

Ou, Sai-Hong Ignatius
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Irvine, Sch Med, Chao Family Comprehens Canc Ctr, Orange, CA 92868 USA South Texas Accelerated Res Therapeut, San Antonio, TX USA
[4]
Molecular Changes Associated with Acquired Resistance to Crizotinib in ROS1-Rearranged Non-Small Cell Lung Cancer
[J].
Song, Ahnah
;
Kim, Tae Min
;
Kim, Dong-Wan
;
Kim, Soyeon
;
Keam, Bhumsuk
;
Lee, Se-Hoon
;
Heo, Dae Seog
.
CLINICAL CANCER RESEARCH,
2015, 21 (10)
:2379-2387

Song, Ahnah
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea

Kim, Tae Min
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea
Seoul Natl Univ Hosp, Dept Internal Med, Seoul 110744, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea

Kim, Dong-Wan
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea
Seoul Natl Univ Hosp, Dept Internal Med, Seoul 110744, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea

Kim, Soyeon
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea

Keam, Bhumsuk
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea
Seoul Natl Univ Hosp, Dept Internal Med, Seoul 110744, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea

Lee, Se-Hoon
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea
Seoul Natl Univ Hosp, Dept Internal Med, Seoul 110744, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea

Heo, Dae Seog
论文数: 0 引用数: 0
h-index: 0
机构:
Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea
Seoul Natl Univ Hosp, Dept Internal Med, Seoul 110744, South Korea Seoul Natl Univ, Coll Med, Canc Res Inst, Seoul, South Korea
[5]
PF-06463922 is a potent and selective next-generation ROS1/ALK inhibitor capable of blocking crizotinib-resistant ROS1 mutations
[J].
Zou, Helen Y.
;
Li, Qiuhua
;
Engstrom, Lars D.
;
West, Melissa
;
Appleman, Vicky
;
Wong, Katy A.
;
McTigue, Michele
;
Deng, Ya-Li
;
Liu, Wei
;
Brooun, Alexei
;
Timofeevski, Sergei
;
McDonnell, Scott R. P.
;
Jiang, Ping
;
Falk, Matthew D.
;
Lappin, Patrick B.
;
Affolter, Timothy
;
Nichols, Tim
;
Hu, Wenyue
;
Lam, Justine
;
Johnson, Ted W.
;
Smeal, Tod
;
Charest, Al
;
Fantin, Valeria R.
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
2015, 112 (11)
:3493-3498

Zou, Helen Y.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Li, Qiuhua
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Engstrom, Lars D.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

West, Melissa
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Appleman, Vicky
论文数: 0 引用数: 0
h-index: 0
机构:
Tufts Med Ctr, Mol Oncol Res Inst, Boston, MA 02111 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Wong, Katy A.
论文数: 0 引用数: 0
h-index: 0
机构:
Tufts Med Ctr, Mol Oncol Res Inst, Boston, MA 02111 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

McTigue, Michele
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Med Chem, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Deng, Ya-Li
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Med Chem, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Liu, Wei
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Med Chem, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Brooun, Alexei
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Med Chem, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Timofeevski, Sergei
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

McDonnell, Scott R. P.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Jiang, Ping
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Falk, Matthew D.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Lappin, Patrick B.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Drug Safety Res & Dev, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Affolter, Timothy
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Drug Safety Res & Dev, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Nichols, Tim
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Drug Safety Res & Dev, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Hu, Wenyue
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Drug Safety Res & Dev, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Lam, Justine
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Pharmacokinet Dynam Metab, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Johnson, Ted W.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Med Chem, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Smeal, Tod
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Charest, Al
论文数: 0 引用数: 0
h-index: 0
机构:
Tufts Med Ctr, Mol Oncol Res Inst, Boston, MA 02111 USA
Tufts Univ, Sch Med, Dept Neurosurg, Boston, MA 02111 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA

Fantin, Valeria R.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA Pfizer Worldwide Res, Oncol Res Unit, La Jolla, CA 92121 USA