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- [1] A phase II study of TAS-117 in patients with advanced solid tumors harboring germline PTEN inactivating mutationsANNALS OF ONCOLOGY, 2021, 32 : S616 - S617Rodon, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USAFunchain, P.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44106 USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USALaetsch, T. W.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Childrens Hosp Philadelphia, Oncol, Philadelphia, PA 19104 USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USASinger, C. F.论文数: 0 引用数: 0 h-index: 0机构: Med Univ Vienna, Womens Univ Clin, Vienna, Austria Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USAArkenau, H-T.论文数: 0 引用数: 0 h-index: 0机构: Inst SCRI UK, SCRI Sarah Cannon Res, London, England Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USAChawla, S. P.论文数: 0 引用数: 0 h-index: 0机构: Southern Calif Santa Mon, Ctr Canc, Sarcoma Oncol Ctr, Santa Monica, CA USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USAHervieu, A.论文数: 0 引用数: 0 h-index: 0机构: Ctr Georges Francois Leclerc Dijon, Med Oncol, Dijon, France Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USAYamamiya, I.论文数: 0 引用数: 0 h-index: 0机构: Bioanalyt DMPK Inc, Taiho Oncol, Princeton, NJ USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USALiu, M.论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol Inc, Biostat, Princeton, NJ USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USABenhadji, K. A.论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol Inc, Clin Dev, Princeton, NJ USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USATakahashi, O.论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol Inc, Clin Dev, Princeton, NJ USA Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USADelaloge, S.论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Med Oncol, Villejuif, France Univ Texas MD Anderson Canc Ctr, Early Drug Dev, Houston, TX 77030 USA
- [2] A phase II study of TAS-117 in patients with advanced solid tumors harboring germline PTEN-inactivating mutationsFUTURE ONCOLOGY, 2022, 18 (30) : 3377 - 3387Rodon, Jordi论文数: 0 引用数: 0 h-index: 0机构: MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAFunchain, Pauline论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Cleveland, OH 44195 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USALaetsch, Theodore W.论文数: 0 引用数: 0 h-index: 0机构: Childrens Hosp Philadelphia, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAArkenau, Hendrik-Tobias论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, London, England UCL, Canc Inst, London W1G 6AD, England MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAHervieu, Alice论文数: 0 引用数: 0 h-index: 0机构: Ctr Georges Francois Leclerc, Dijon, France MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USASinger, Christian F.论文数: 0 引用数: 0 h-index: 0机构: Med Univ Vienna, Dept OB GYN, A-1090 Vienna, Austria Med Univ Vienna, Comprehens Canc Ctr, A-1090 Vienna, Austria MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAMurciano-Goroff, Yonina R.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10065 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAChawla, Sant P.论文数: 0 引用数: 0 h-index: 0机构: Sarcoma Oncol Res Ctr, Santa Monica, CA 90403 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAAnthony, Kristin论文数: 0 引用数: 0 h-index: 0机构: PTEN Hamartoma Tumor Syndrome Fdn, Huntsville, AL 35806 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAYamamiya, Ikuo论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol, Princeton, NJ 08540 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USALiu, Mei论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol, Princeton, NJ 08540 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USAHalim, Abdel-Baset论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol, Princeton, NJ 08540 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USABenhadji, Karim A.论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol, Princeton, NJ 08540 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USATakahashi, Osamu论文数: 0 引用数: 0 h-index: 0机构: Taiho Oncol, Princeton, NJ 08540 USA MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USADelaloge, Suzette论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, F-94805 Villejuif, France MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Div Canc Med, Houston, TX 77030 USA
- [3] A first-in-human phase I study of TAS-117, an allosteric AKT inhibitor, in patients with advanced solid tumorsCANCER CHEMOTHERAPY AND PHARMACOLOGY, 2024, 93 (06) : 605 - 616Doi, Toshihiko论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanTakahashi, Shunji论文数: 0 引用数: 0 h-index: 0机构: Canc Inst Hosp, Japanese Fdn Canc Res, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanAoki, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Keio Univ, Sch Med, Tokyo, Japan Akasaka Sannou Med Ctr, Tokyo, Japan Int Univ Hlth & Welf, Grad Sch, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanYonemori, Kan论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHara, Hiroki论文数: 0 引用数: 0 h-index: 0机构: Saitama Canc Ctr, Kita Adachi, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHasegawa, Kosei论文数: 0 引用数: 0 h-index: 0机构: Saitama Med Univ, Int Med Ctr, Hidaka, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanTakehara, Kazuhiro论文数: 0 引用数: 0 h-index: 0机构: NHO Shikoku Canc Ctr, Matsuyama, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHarano, Kenichi论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanYunokawa, Mayu论文数: 0 引用数: 0 h-index: 0机构: Canc Inst Hosp, Japanese Fdn Canc Res, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, Japan论文数: 引用数: h-index:机构:Shimoi, Tatsunori论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHorie, Koji论文数: 0 引用数: 0 h-index: 0机构: Saitama Canc Ctr, Kita Adachi, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanOgasawara, Aiko论文数: 0 引用数: 0 h-index: 0机构: Saitama Med Univ, Int Med Ctr, Hidaka, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanOkame, Shinichi论文数: 0 引用数: 0 h-index: 0机构: NHO Shikoku Canc Ctr, Matsuyama, Japan Natl Canc Ctr Hosp East, Kashiwa, Japan
- [4] Dose escalation of tinostamustine in patients with advanced solid tumorsCANCER RESEARCH, 2019, 79 (13)Mita, Alain论文数: 0 引用数: 0 h-index: 0机构: Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA Cedars Sinai Med Ctr, Los Angeles, CA 90048 USALoeffler, Markus论文数: 0 引用数: 0 h-index: 0机构: Mundipharma EDO GmbH EDO, Basel, Switzerland Cedars Sinai Med Ctr, Los Angeles, CA 90048 USABui, Nam论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Stanford Canc Inst, Stanford, CA 94305 USA Cedars Sinai Med Ctr, Los Angeles, CA 90048 USAMehrling, Thomas论文数: 0 引用数: 0 h-index: 0机构: Mundipharma EDO GmbH EDO, Basel, Switzerland Cedars Sinai Med Ctr, Los Angeles, CA 90048 USARimmel, Bobbie J.论文数: 0 引用数: 0 h-index: 0机构: Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA Cedars Sinai Med Ctr, Los Angeles, CA 90048 USANatale, Ronald B.论文数: 0 引用数: 0 h-index: 0机构: Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA Cedars Sinai Med Ctr, Los Angeles, CA 90048 USAKummar, Shivaani论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Stanford Canc Inst, Stanford, CA 94305 USA Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA
- [5] First-in-human phase I study of TAS-117, an allosteric AKT inhibitor, in patients with advanced solid tumoursANNALS OF ONCOLOGY, 2019, 30Yunokawa, M.论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanTakahashi, S.论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanAoki, D.论文数: 0 引用数: 0 h-index: 0机构: Keio Univ Hosp, Dept Obstet & Gynecol, Tokyo, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanYonemori, K.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Dept Breast & Med Oncol, Tokyo, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanHara, H.论文数: 0 引用数: 0 h-index: 0机构: Saitama Canc Ctr, Dept Gastroenterol, Saitama, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanHasegawa, K.论文数: 0 引用数: 0 h-index: 0机构: Saitama Med Univ, Int Med Ctr, Dept Gynecol Oncol, Saitama, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanTakehara, K.论文数: 0 引用数: 0 h-index: 0机构: Natl Hosp Org Shikoku Canc Ctr, Dept Gynecol Oncol, Matsuyama, Ehime, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanHarano, K.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Dept Expt Therapeut, Chiba, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanNomura, H.论文数: 0 引用数: 0 h-index: 0机构: Keio Univ Hosp, Dept Obstet & Gynecol, Tokyo, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanNoguchi, E.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Dept Breast & Med Oncol, Tokyo, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanHorie, K.论文数: 0 引用数: 0 h-index: 0机构: Saitama Canc Ctr, Depertment Gynecol, Saitama, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanOgasawara, A.论文数: 0 引用数: 0 h-index: 0机构: Saitama Med Univ, Int Med Ctr, Dept Gynecol Oncol, Saitama, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanOkame, S.论文数: 0 引用数: 0 h-index: 0机构: Natl Hosp Org Shikoku Canc Ctr, Dept Gynecol Oncol, Matsuyama, Ehime, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, JapanDoi, T.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Dept Expt Therapeut, Chiba, Japan Japanese Fdn Canc Res, Dept Med Oncol, Canc Inst Hosp, Tokyo, Japan
- [6] A dose escalation study of weekly docetaxel in patients with advanced solid tumorsCANCER CHEMOTHERAPY AND PHARMACOLOGY, 2000, 46 (06) : 488 - 492Kouroussis, C论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceAgelaki, S论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceMavroudis, D论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceSouglakos, J论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceKakolyris, S论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceKalbakis, K论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceVardakis, N论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceReppa, D论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceHatzidaki, D论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceSamonis, G论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, GreeceGeorgoulias, V论文数: 0 引用数: 0 h-index: 0机构: Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece Univ Gen Hosp Heraklion, Dept Med Oncol, GR-71110 Crete, Greece
- [7] A dose escalation study of weekly docetaxel in patients with advanced solid tumorsCancer Chemotherapy and Pharmacology, 2000, 46 : 488 - 492Ch. Kouroussis论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,S. Agelaki论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,D. Mavroudis论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,J. Souglakos论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,S. Kakolyris论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,K. Kalbakis论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,N. Vardakis论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,D. Reppa论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,D. Hatzidaki论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,G. Samonis论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,V. Georgoulias论文数: 0 引用数: 0 h-index: 0机构: Department of Medical Oncology,
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- [10] Phase I dose escalation trial of pegzilarginase in patients with advanced solid tumorsCANCER RESEARCH, 2018, 78 (13)Rasco, Drew W.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, San Antonio, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USAEckhardt, S. Gail论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Sch Med, Denver, CO USA South Texas Accelerated Res Therapeut, San Antonio, TX USADavar, Diwakar论文数: 0 引用数: 0 h-index: 0机构: Univ Pittsburgh, Pittsburgh, PA USA South Texas Accelerated Res Therapeut, San Antonio, TX USALewis, Karl论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Sch Med, Denver, CO USA South Texas Accelerated Res Therapeut, San Antonio, TX USALara-Guerra, Humberto论文数: 0 引用数: 0 h-index: 0机构: Aeglea Biotherapeut, Austin, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USAAlters, Susan E.论文数: 0 引用数: 0 h-index: 0机构: Aeglea Biotherapeut, Austin, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USAEckert, Stephen论文数: 0 引用数: 0 h-index: 0机构: Aeglea Biotherapeut, Austin, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USARowlinson, Scott W.论文数: 0 引用数: 0 h-index: 0机构: Aeglea Biotherapeut, Austin, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USAWooldridge, James E.论文数: 0 引用数: 0 h-index: 0机构: Aeglea Biotherapeut, Austin, TX USA South Texas Accelerated Res Therapeut, San Antonio, TX USACarvajal, Richard D.论文数: 0 引用数: 0 h-index: 0机构: Herbert Irving Comprehens Canc Ctr, New York, NY USA South Texas Accelerated Res Therapeut, San Antonio, TX USA