Condensed bridgehead nitrogen heterocyclic systems:: Facile synthesis and antimicrobial activity of imidazo [2,1-b]-1,3,4-thiadiazoles

被引：0

作者：

Mohan, J ^{[1
]}

Kumar, A ^{[1
]}

机构：

[1] Maharshi Dayanand Univ, Dept Chem, Rohtak 124001, Haryana, India

来源：

INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2003年 / 13卷 / 02期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of 2,6-diarylimidazo [2,1-b]-1,3,4-thiadiazoles 2 has been achieved by the reaction of alpha-haloketones with 2-amino-5-(2-pyridyl)-1,3,4-thiadiazole 1 or more conveniently by treating I directly with ketones in presence of NBS. Bromination of 2 furnished 5-bromo-2,6-diarylimidazo [2,1-b]-1,3,4-thiadiazoles 3. The antimicrobial activity of some of the compounds has been evaluated.

引用

页码：101 / 104

页数：4

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