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Steroid sulfatase inhibitors: from concept to clinic
被引:0
作者
:
Potter, B. V. L.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Bath BA2 7AY, Avon, England
Univ Bath, Bath BA2 7AY, Avon, England
Potter, B. V. L.
[
1
]
机构
:
[1]
Univ Bath, Bath BA2 7AY, Avon, England
来源
:
JOURNAL OF PHARMACY AND PHARMACOLOGY
|
2007年
/ 59卷
关键词
:
D O I
:
暂无
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
210
引用
收藏
页码:A76 / A76
页数:1
相关论文
共 6 条
[1]
ESTRONE SULFAMATES - POTENT INHIBITORS OF ESTRONE SULFATASE WITH THERAPEUTIC POTENTIAL
HOWARTH, NM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
HOWARTH, NM
PUROHIT, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
PUROHIT, A
REED, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
REED, MJ
POTTER, BVL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
POTTER, BVL
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1994,
37
(02)
: 219
-
221
[2]
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: Synthesis, in vitro SAR, protein crystallography, and in vivo activity
Leese, Mathew P.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Leese, Mathew P.
Leblond, Bertrand
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Leblond, Bertrand
Smith, Andrew
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Smith, Andrew
Newman, Simon P.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Newman, Simon P.
Di Fiore, Anna
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Di Fiore, Anna
De Simone, Giuseppina
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
De Simone, Giuseppina
Supuran, Claudiu T.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Supuran, Claudiu T.
Purohit, Atul
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Purohit, Atul
Reed, Michael J.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Reed, Michael J.
Potter, Barry V. L.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Potter, Barry V. L.
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
2006,
49
(26)
: 7683
-
7696
[3]
Crystal structure of human carbonic anhydrase II at 1.95 Å resolution in complex with 667-cournate, a novel anti-cancer agent
Lloyd, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Lloyd, MD
Pederick, RL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Pederick, RL
Natesh, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Natesh, R
Woo, LWL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Woo, LWL
Purohit, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Purohit, A
Reed, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Reed, MJ
Acharya, KR
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Acharya, KR
Potter, NL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Potter, NL
[J].
BIOCHEMICAL JOURNAL,
2005,
385
: 715
-
720
[4]
Phase I study of STX 64 (667 Coumate) in breast cancer patients: The first study of a steroid sulfatase inhibitor
Stanway, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Stanway, SJ
Purohit, A
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Purohit, A
Woo, LWL
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Woo, LWL
Sufi, S
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Sufi, S
Vigushin, D
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Vigushin, D
Ward, R
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Ward, R
Wilson, RH
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Wilson, RH
Stanczyk, FZ
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Stanczyk, FZ
Dobbs, N
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Dobbs, N
Kulinskaya, E
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Kulinskaya, E
Elliott, M
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Elliott, M
Potter, BVL
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Potter, BVL
Reed, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Reed, MJ
Coombes, RC
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Coombes, RC
[J].
CLINICAL CANCER RESEARCH,
2006,
12
(05)
: 1585
-
1592
[5]
Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates
Woo, LWL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Woo, LWL
Purohit, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Purohit, A
Malini, B
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Malini, B
Reed, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Reed, MJ
Potter, BVL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Potter, BVL
[J].
CHEMISTRY & BIOLOGY,
2000,
7
(10):
: 773
-
791
[6]
WOO LWL, 2007, IN PRESS J MED CHEM
←
1
→
共 6 条
[1]
ESTRONE SULFAMATES - POTENT INHIBITORS OF ESTRONE SULFATASE WITH THERAPEUTIC POTENTIAL
HOWARTH, NM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
HOWARTH, NM
PUROHIT, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
PUROHIT, A
REED, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
REED, MJ
POTTER, BVL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV BATH,SCH PHARM & PHARMACOL,DEPT MED CHEM,BATH BA2 7AY,AVON,ENGLAND
POTTER, BVL
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1994,
37
(02)
: 219
-
221
[2]
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: Synthesis, in vitro SAR, protein crystallography, and in vivo activity
Leese, Mathew P.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Leese, Mathew P.
Leblond, Bertrand
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Leblond, Bertrand
Smith, Andrew
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Smith, Andrew
Newman, Simon P.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Newman, Simon P.
Di Fiore, Anna
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Di Fiore, Anna
De Simone, Giuseppina
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
De Simone, Giuseppina
Supuran, Claudiu T.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Supuran, Claudiu T.
Purohit, Atul
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Purohit, Atul
Reed, Michael J.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Reed, Michael J.
Potter, Barry V. L.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Potter, Barry V. L.
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
2006,
49
(26)
: 7683
-
7696
[3]
Crystal structure of human carbonic anhydrase II at 1.95 Å resolution in complex with 667-cournate, a novel anti-cancer agent
Lloyd, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Lloyd, MD
Pederick, RL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Pederick, RL
Natesh, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Natesh, R
Woo, LWL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Woo, LWL
Purohit, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Purohit, A
Reed, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Reed, MJ
Acharya, KR
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Acharya, KR
Potter, NL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Sterix Ltd, Bath BA2 7AY, Avon, England
Potter, NL
[J].
BIOCHEMICAL JOURNAL,
2005,
385
: 715
-
720
[4]
Phase I study of STX 64 (667 Coumate) in breast cancer patients: The first study of a steroid sulfatase inhibitor
Stanway, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Stanway, SJ
Purohit, A
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Purohit, A
Woo, LWL
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Woo, LWL
Sufi, S
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Sufi, S
Vigushin, D
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Vigushin, D
Ward, R
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Ward, R
Wilson, RH
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Wilson, RH
Stanczyk, FZ
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Stanczyk, FZ
Dobbs, N
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Dobbs, N
Kulinskaya, E
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Kulinskaya, E
Elliott, M
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Elliott, M
Potter, BVL
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Potter, BVL
Reed, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Reed, MJ
Coombes, RC
论文数:
0
引用数:
0
h-index:
0
机构:
St Marys Hosp, Imperial Coll, Fac Med, Endocrinol & Metab Med & Sterix Ltd, London W2 1NY, England
Coombes, RC
[J].
CLINICAL CANCER RESEARCH,
2006,
12
(05)
: 1585
-
1592
[5]
Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates
Woo, LWL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Woo, LWL
Purohit, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Purohit, A
Malini, B
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Malini, B
Reed, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Reed, MJ
Potter, BVL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Univ Bath, Dept Pharm & Pharmacol, Bath BA2 7AY, Avon, England
Potter, BVL
[J].
CHEMISTRY & BIOLOGY,
2000,
7
(10):
: 773
-
791
[6]
WOO LWL, 2007, IN PRESS J MED CHEM
←
1
→