A Highly Efficient Bismuth Salts-Catalyzed Route for the Synthesis of α-Aminophosphonates

被引：29

作者：

Banik, Antara ^{[1
]}

Batta, Sahil ^{[1
]}

Bandyopadhyay, Debasish ^{[1
]}

Banik, Bimal K. ^{[1
]}

机构：

[1] Univ Texas Pan Amer, Dept Chem, Edinburg, TX 78541 USA

来源：

MOLECULES | 2010年 / 15卷 / 11期

关键词：

bismuth salts; catalysis; imines; phosphites; alpha-aminophosphonates; ONE-POT SYNTHESIS; POLYCYCLIC AROMATIC-COMPOUNDS; ANTICANCER BETA-LACTAMS; SOLVENT-FREE CONDITIONS; AMINO PHOSPHONATES; BIOLOGICAL EVALUATION; MICHAEL REACTIONS; ROOM-TEMPERATURE; NITRATE; AGENTS;

D O I：

10.3390/molecules15118205

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

A convenient synthesis of different types of alpha-amino phosphonates via one-pot solvent-free three component reactions of aldehydes, amines and phosphites catalyzed by bismuth salts has been investigated. Bismuth triflate is found to be the most effective catalyst for this reaction.

引用

页码：8205 / 8213

页数：9

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