Synthesis of 1-arylsulfonyl-3-N-(β-D-methyl acetylglucuronate-1-yl)-5-fluorouracil

被引：1
|
作者：
Zhou, FY
Sun, CJ [1 ]
Li, JH
机构：
[1] Zaozhuang Normal Coll, Dept Chem, Shandong 277160, Zaozhuang, Peoples R China
[2] Shandong Univ, Dept Chem, Jinan 250100, Peoples R China
来源：
SYNTHETIC COMMUNICATIONS | 2001年 / 31卷 / 18期
关键词：
D O I：
10.1081/SCC-100105334
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Five glucuronides of 1-arylsulfonyl-5-fluorouracil were synthesized by the reaction of 1-arylsulfonyl-5-fluorouracil 2 with methyl 2,3,4-tri-O-acetyl-1-bromo-1-deoxy-alpha -D-glucuronate I under phase transfer catalysis. Their structures were confirmed by IR, H-1 NMR and elementary analysis.
引用
收藏
页码：2837 / 2840
页数：4
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