Triazolopyridazine derivatives as selective and orally bioavailable c-Met inhibitors

被引:0
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作者
Romero, Karina [1 ]
Bauer, David [1 ]
Bellon, Steve [2 ]
Berry, Loren M. [3 ]
Bode, Christiane [1 ]
Boezio, Alessandro [1 ]
Broome, Martin [4 ]
Choquette, Deborah [1 ]
Chen, April [3 ]
Dussault, Isabelle [4 ]
Huang, Liyue [3 ]
Kaplan-Lefko, Paula [4 ]
Lewis, Richard [1 ]
Lin, Jasmine [3 ]
Lohman, Julia [1 ]
Potashman, Michele [1 ]
Rex, Karen [4 ]
Shah, Kavitah [5 ]
Shimanovich, Roman [5 ]
Teffera, Yohannes [3 ]
Yang, Yajing [4 ]
Zhang, Michael [4 ]
Zhao, Zhiyang [4 ]
Harmange, Jean-Claude [1 ]
机构
[1] Amgen Inc, Dept Med Chem, Cambridge, MA 02139 USA
[2] Amgen Inc, Dept Mol Struct, Cambridge, MA 02139 USA
[3] Amgen Inc, Dept Pharmacokinet & Drug Metab, Cambridge, MA 02139 USA
[4] Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA
[5] Amgen Inc, Dept Small Mol Prod Dev, Cambridge, MA 02139 USA
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2009年 / 238卷
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
136-MEDI
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页数:1
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