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- [1] Discovery and optimization of potent and selective triazolopyridazine series of c-Met inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (22) : 6307 - 6312Boezio, Alessandro A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USABerry, Loren论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAAlbrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USABauer, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USABellon, Steven F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USABode, Christiane论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAChen, April论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAChoquette, Deborah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USADussault, Isabelle论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAHirai, Satoko论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAKaplan-Lefko, Paula论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USALarrow, Jay F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USALin, Min-Hwa Jasmine论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USALohman, Julia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAPotashman, Michele H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USARex, Karen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USASantostefano, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAShah, Kavita论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAShimanovich, Roman论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USASpringer, Stephanie K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USATeffera, Yohannes论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAZhang, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAHarmange, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA
- [2] Selective and Orally Bioavailable c-Met PROTACs for the Treatment of c-Met-Addicted CancerJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (19) : 17053 - 17069Ying, Shilong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaChi, Hongli论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaWu, Xiaoqiu论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaZeng, Pingping论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ Technol, Coll Mat Sci & Engn, Hangzhou 310014, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaChen, Jinling论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaFu, Ting论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaFu, Weitao论文数: 0 引用数: 0 h-index: 0机构: Hefei Comprehens Natl Sci Ctr, Insitute Hlth & Med, Hefei 230601, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaZhang, Penghui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R ChinaTan, Weihong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China Shanghai Jiao Tong Univ, Renji Hosp, Inst Mol Med, Sch Med, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Coll Chem & Chem Engn, Shanghai 200240, Peoples R China Chinese Acad Sci, Zhejiang Canc Hosp, Hangzhou Inst Med HIM, Key Lab Zhejiang Prov Aptamers & Theranost, Hangzhou 310022, Zhejiang, Peoples R China
- [3] Discovery and optimization of potent and selective triazolopyridazine series of c-Met inhibitors (vol 19, pg 6307, 2009)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (02) : 773 - 773Boezio, Alessandro A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USABerry, Loren论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAAlbrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USABauer, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USABellon, Steven F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USABode, Christiane论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAChen, April论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAChoquette, Deborah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USADussault, Isabelle论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAFang, Mei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAHirai, Satoko论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAKaplan-Lefko, Paula论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USALarrow, Jay F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USALin, Min-Hwa Jasmine论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USALohman, Julia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAPotashman, Michele H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAQu, Yusheng论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USARex, Karen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USASantostefano, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAShah, Kavita论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAShimanovich, Roman论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USASpringer, Stephanie K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USATeffera, Yohannes论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAZhang, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USAHarmange, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA
- [4] Triazolopyridazine derivatives: Synthesis, cytotoxic evaluation, c-Met kinase activity and molecular dockingBIOORGANIC CHEMISTRY, 2019, 92Ahmed, Eman M.论文数: 0 引用数: 0 h-index: 0机构: Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, Egypt Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, EgyptKhalil, Nadia A.论文数: 0 引用数: 0 h-index: 0机构: Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, Egypt Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, EgyptTaher, Azza T.论文数: 0 引用数: 0 h-index: 0机构: Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, Egypt October 6 Univ, Pharmaceut Organ Chem Dept, Fac Pharm, Giza, Egypt Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, EgyptRefaey, Rana H.论文数: 0 引用数: 0 h-index: 0机构: October Univ Modern Sci & Arts MSA, Pharmaceut Chem Dept, Fac Pharm, Giza, Egypt Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, EgyptNissan, Yassin M.论文数: 0 引用数: 0 h-index: 0机构: October Univ Modern Sci & Arts MSA, Pharmaceut Chem Dept, Fac Pharm, Giza, Egypt Cairo Univ, Pharmaceut Chem Dept, Fac Pharm, Kasr Elini St, Cairo 11562, Egypt Cairo Univ, Fac Pharm, Pharmaceut Organ Chem Dept, Cairo, Egypt
- [5] Synthesis of triazolotriazine derivatives as c-Met inhibitorsMolecular Diversity, 2021, 25 : 839 - 846Yuting Guo论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryXia Peng论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryYinchun Ji论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryYitong Zhang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryJian Ding论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryZhengsheng Zhan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryJing Ai论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal ChemistryWenhu Duan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Institute of Materia Medica,Department of Medicinal Chemistry
- [6] Synthesis of triazolotriazine derivatives as c-Met inhibitorsMOLECULAR DIVERSITY, 2021, 25 (02) : 839 - 846Guo, Yuting论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaPeng, Xia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaJi, Yinchun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaZhang, Yitong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaDing, Jian论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaZhan, Zhengsheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaAi, Jing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R ChinaDuan, Wenhu论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China
- [7] Identification of orally active small molecule c-met inhibitorsCANCER RESEARCH, 2009, 69Miknyoczki, Sheila论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAUnderiner, Ted论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAAimone, Lisa论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAChang, Hong论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAGalinis, Debbie论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAGrobelny, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAHebertz, Torsten论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAHuang, Zeqi论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAHusten, Jean论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAMikiewicz, Karen论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAMurthy, Seetha论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAPritchard, Sonya论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAWeinberg, Linda论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAWorrell, Candace论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USAAtor, Mark论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USADorsey, Bruce论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USARuggeri, Bruce论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, W Chester, PA USA Cephalon Inc, W Chester, PA USA
- [8] c-Met inhibitorsINFECTIOUS AGENTS AND CANCER, 2013, 8Mughal, Anum论文数: 0 引用数: 0 h-index: 0机构: Dow Univ Hlth Sci, Dow Med Coll, Karachi, Pakistan Dow Univ Hlth Sci, Dow Med Coll, Karachi, PakistanAslam, Hafiz Muhammad论文数: 0 引用数: 0 h-index: 0机构: Dow Univ Hlth Sci, Dow Med Coll, Karachi, Pakistan Dow Univ Hlth Sci, Dow Med Coll, Karachi, PakistanSheikh, Asfandyar论文数: 0 引用数: 0 h-index: 0机构: Dow Univ Hlth Sci, Dow Med Coll, Karachi, Pakistan Pakistan Res Evolut Students Soc, Karachi, Pakistan Dow Univ Hlth Sci, Dow Med Coll, Karachi, PakistanKhan, Agha Muhammad Hammad论文数: 0 引用数: 0 h-index: 0机构: Dow Univ Hlth Sci, Sindh Med Coll, Karachi, Pakistan Dow Univ Hlth Sci, Dow Med Coll, Karachi, PakistanSaleem, Shafaq论文数: 0 引用数: 0 h-index: 0机构: Dow Univ Hlth Sci, Dow Med Coll, Karachi, Pakistan Dow Univ Hlth Sci, Dow Med Coll, Karachi, Pakistan
- [9] C-MET INHIBITORSJOURNAL OF THORACIC ONCOLOGY, 2012, 7 (06) : S22 - S22Adjei, A. A.论文数: 0 引用数: 0 h-index: 0机构: Roswell Pk Canc Inst, Dept Med, Buffalo, NY 14263 USA Roswell Pk Canc Inst, Dept Med, Buffalo, NY 14263 USA
- [10] c-Met inhibitorsInfectious Agents and Cancer, 8Anum Mughal论文数: 0 引用数: 0 h-index: 0机构: Dow University of Health Sciences,Dow Medical CollegeHafiz Muhammad Aslam论文数: 0 引用数: 0 h-index: 0机构: Dow University of Health Sciences,Dow Medical CollegeAsfandyar Sheikh论文数: 0 引用数: 0 h-index: 0机构: Dow University of Health Sciences,Dow Medical CollegeAgha Muhammad Hammad Khan论文数: 0 引用数: 0 h-index: 0机构: Dow University of Health Sciences,Dow Medical CollegeShafaq Saleem论文数: 0 引用数: 0 h-index: 0机构: Dow University of Health Sciences,Dow Medical College