共 65 条
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(R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells
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Barsyte-Lovejoy, Dalia
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Li, Fengling
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Oudhoff, Menno J.
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Tatlock, John H.
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Dong, Aiping
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Zeng, Hong
;
Wu, Hong
;
Freeman, Spencer A.
;
Schapira, Matthieu
;
Senisterra, Guillermo A.
;
Kuznetsova, Ekaterina
;
Marcellus, Richard
;
Allali-Hassani, Abdellah
;
Kennedy, Steven
;
Lambert, Jean-Philippe
;
Couzens, Amber L.
;
Aman, Ahmed
;
Gingras, Anne-Claude
;
Al-Awar, Rima
;
Fish, Paul V.
;
Gerstenberger, Brian S.
;
Roberts, Lee
;
Benn, Caroline L.
;
Grimley, Rachel L.
;
Braam, Mitchell J. S.
;
Rossi, Fabio M. V.
;
Sudol, Marius
;
Brown, Peter J.
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Bunnage, Mark E.
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Owen, Dafydd R.
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Zaph, Colby
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Vedadi, Masoud
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Arrowsmith, Cheryl H.
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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
2014, 111 (35)
:12853-12858

Barsyte-Lovejoy, Dalia
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Li, Fengling
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Oudhoff, Menno J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ British Columbia, Biomed Res Ctr, Vancouver, BC V6T 1Z3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Tatlock, John H.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Dong, Aiping
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Zeng, Hong
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Wu, Hong
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Freeman, Spencer A.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ British Columbia, Dept Microbiol & Immunol, Vancouver, BC V6T 1Z3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

论文数: 引用数:
h-index:
机构:

Senisterra, Guillermo A.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Kuznetsova, Ekaterina
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Marcellus, Richard
论文数: 0 引用数: 0
h-index: 0
机构:
Ontario Inst Canc Res, Drug Discovery Program, Toronto, ON M5G 0A3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Allali-Hassani, Abdellah
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Kennedy, Steven
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Lambert, Jean-Philippe
论文数: 0 引用数: 0
h-index: 0
机构:
Lunenfeld Tanenbaum Res Inst, Ctr Syst Biol, Toronto, ON M5G 1X5, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Couzens, Amber L.
论文数: 0 引用数: 0
h-index: 0
机构:
Lunenfeld Tanenbaum Res Inst, Ctr Syst Biol, Toronto, ON M5G 1X5, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Aman, Ahmed
论文数: 0 引用数: 0
h-index: 0
机构:
Ontario Inst Canc Res, Drug Discovery Program, Toronto, ON M5G 0A3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Gingras, Anne-Claude
论文数: 0 引用数: 0
h-index: 0
机构:
Lunenfeld Tanenbaum Res Inst, Ctr Syst Biol, Toronto, ON M5G 1X5, Canada
Univ Toronto, Dept Mol Genet, Toronto, ON M5S 1A8, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Al-Awar, Rima
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Dept Pharmacol & Toxicol, Toronto, ON M5S 1A8, Canada
Ontario Inst Canc Res, Drug Discovery Program, Toronto, ON M5G 0A3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Fish, Paul V.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Worldwide Med Chem, Sandwich CT13 9NJ, Kent, England Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Gerstenberger, Brian S.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Worldwide Med Chem, Groton, CT 06340 USA Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Roberts, Lee
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Worldwide Med Chem, Cambridge, MA 02139 USA Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Benn, Caroline L.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Neusentis Res Unit, Cambridge CB21 6GS, England Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Grimley, Rachel L.
论文数: 0 引用数: 0
h-index: 0
机构: Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Braam, Mitchell J. S.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ British Columbia, Biomed Res Ctr, Vancouver, BC V6T 1Z3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Rossi, Fabio M. V.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ British Columbia, Biomed Res Ctr, Vancouver, BC V6T 1Z3, Canada
Univ British Columbia, Dept Med Genet, Vancouver, BC V6T 1Z3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Sudol, Marius
论文数: 0 引用数: 0
h-index: 0
机构:
Geisinger Med Clin, Weis Ctr Res, Danville, PA 17821 USA Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Brown, Peter J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Bunnage, Mark E.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Worldwide Med Chem, Cambridge, MA 02139 USA Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Owen, Dafydd R.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Worldwide Med Chem, Cambridge, MA 02139 USA Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Zaph, Colby
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h-index: 0
机构:
Univ British Columbia, Biomed Res Ctr, Vancouver, BC V6T 1Z3, Canada
Univ British Columbia, Dept Pathol & Lab Med, Vancouver, BC V6T 1Z3, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Vedadi, Masoud
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
Univ Toronto, Dept Pharmacol & Toxicol, Toronto, ON M5S 1A8, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Arrowsmith, Cheryl H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
Univ Toronto, Princess Margaret Canc Ctr, Toronto, ON M5G 1L7, Canada
Univ Toronto, Dept Med Biophys, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
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Ben-David, Uri
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h-index: 0
机构:
Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Weissbein, Uri
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h-index: 0
机构:
Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Mandefro, Berhan
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h-index: 0
机构:
Cedars Sinai Med Ctr, Dept Biomed Sci, Los Angeles, CA 90048 USA
Cedars Sinai Med Ctr, Regenerat Med Inst, Los Angeles, CA 90048 USA Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Maimon, Adva
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h-index: 0
机构:
Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Golan-Lev, Tamar
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h-index: 0
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Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Narwani, Kavita
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h-index: 0
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Cedars Sinai Med Ctr, Dept Biomed Sci, Los Angeles, CA 90048 USA
Cedars Sinai Med Ctr, Regenerat Med Inst, Los Angeles, CA 90048 USA Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Clark, Amander T.
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h-index: 0
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Univ Calif Los Angeles, Dept Mol Cell & Dev Biol, Los Angeles, CA 90095 USA
Univ Calif Los Angeles, Eli & Edythe Broad Ctr Regenerat Med & Stem Cell, Los Angeles, CA 90095 USA Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Andrews, Peter W.
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Univ Sheffield, Dept Biomed Sci, Ctr Stem Cell Biol, Sheffield S10 2TN, S Yorkshire, England Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Benvenisty, Nissim
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Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel

Biancotti, Juan Carlos
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Cedars Sinai Med Ctr, Dept Biomed Sci, Los Angeles, CA 90048 USA
Cedars Sinai Med Ctr, Regenerat Med Inst, Los Angeles, CA 90048 USA
Univ So Calif, Keck Sch Med, Dept Physiol & Biophys, Zilkha Neurogenet Inst, Los Angeles, CA 90033 USA Hebrew Univ Jerusalem, Silberman Inst Life Sci, Dept Genet, Stem Cell Unit, IL-91904 Jerusalem, Israel
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Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain

Ligero, Gertru
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Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain

Sanchez, Laura
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Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain

de la Cueva, Teresa
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Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain

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Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain

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Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain Univ Granada, Andalusian Stem Cell Bank, Inst Invest Biomed, Granada, Spain