Synthesis of camptothecin-amino acid carbamate linkers

被引：3
作者：
Etienne, Marcus A. [1 ]
Kostochka, Mikhail [1 ]
Fuselier, Joseph A. [1 ]
Coy, David H. [1 ]
机构：
[1] Tulane Univ, Sch Med, Dept Med, Peptide Res Labs,Tulane Hlth Sci Ctr, New Orleans, LA 70112 USA
来源：
AMINO ACIDS | 2012年 / 42卷 / 05期
关键词：
Camptothecin; Somatostatin; Bioconjugates; Amino acids; Linkers; CYCLIZATION-ACTIVATED PRODRUGS; DESIGN; DERIVATIVES; STRATEGIES; RECEPTORS; GROWTH;
D O I：
10.1007/s00726-011-0884-4
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
A more convenient and facile approach for the synthesis and production of camptothecin-amino acids carbamate linkers, that can be used in the synthesis of bioconjugate peptides JF-10-81, JF-10-71, and other peptide analogs designed to target somatostatin receptors has been described.
引用
收藏
页码：1727 / 1733
页数：7
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