Spironolactone and canrenoic acid block hKv1.5 channels

被引:0
|
作者
Caballero, R [1 ]
Gomez, R [1 ]
Nuñez, L [1 ]
Gonzalez, T [1 ]
Arias, C [1 ]
Guizy, M [1 ]
Valenzuela, C [1 ]
Tamargo, J [1 ]
Delpon, E [1 ]
机构
[1] Univ Complutense Madrid, Dept Pharmacol, Sch Med, Madrid, Spain
关键词
D O I
暂无
中图分类号
Q6 [生物物理学];
学科分类号
071011 ;
摘要
引用
收藏
页码:533A / 534A
页数:2
相关论文
共 50 条
  • [1] Spironolactone and canrenoic acid block hKv1.5, Kv4.3 and KvLQT1+minK channels
    Caballero, R
    Gómez, R
    Núñez, L
    Delpón, E
    Tamargo, J
    EUROPEAN HEART JOURNAL, 2004, 25 : 629 - 629
  • [2] Spironolactone and its main metabolite canrenoic acid block hKv1.5, Kv4.3 and Kv7.1+minK channels
    Gómez, R
    Núñez, L
    Caballero, R
    Vaquero, M
    Tamargo, J
    Delpón, E
    BRITISH JOURNAL OF PHARMACOLOGY, 2005, 146 (01) : 146 - 161
  • [3] Nifedipine block of hKv1.5 channels.
    Zhang, X
    Anderson, J
    Fedida, D
    BIOPHYSICAL JOURNAL, 1997, 72 (02) : TUP11 - TUP11
  • [4] Molecular determinants of stereoselective bupivacaine block of hKv1.5 channels
    Franqueza, L
    Longobardo, M
    Vicente, J
    Delpon, E
    Tamkun, MM
    Tamargo, J
    Snyders, DJ
    Valenzuela, C
    CIRCULATION RESEARCH, 1997, 81 (06) : 1053 - 1064
  • [5] Effects of benzocaine on hKv1.5 channels.
    Delpón, E
    Caballero, R
    Valenzuela, C
    Longobardo, M
    Snyders, D
    Tamargo, J
    BIOPHYSICAL JOURNAL, 1998, 74 (02) : A212 - A212
  • [6] Threonine 505 determines stereoselective bupivacaine block of hKv1.5 channels.
    Vicente, J
    Franqueza, L
    Delpon, E
    Tamkun, MM
    Tamargo, J
    Snyders, DJ
    Valenzuela, C
    BIOPHYSICAL JOURNAL, 1997, 72 (02) : TUP10 - TUP10
  • [7] Chemical determinants of stereoselective local anesthetics block of hKv1.5 channels.
    Longobardo, M
    Caballero, R
    Delpón, E
    Tamargo, J
    Valenzuela, C
    BIOPHYSICAL JOURNAL, 1998, 74 (02) : A211 - A211
  • [8] Assembly with the Kvβ1.3 subunit modulates drug block of hKv1.5 channels
    González, T
    Navarro-Polanco, R
    Arias, C
    Caballero, R
    Moreno, I
    Delpón, E
    Tamargo, J
    Tamkun, MM
    Valenzuela, C
    MOLECULAR PHARMACOLOGY, 2002, 62 (06) : 1456 - 1463
  • [9] Evidences for an external bupivacaine receptor in hKv1.5 channels
    Longobardo, M
    Navarro-Polanco, R
    Caballero, R
    Delpon, E
    Tamargo, J
    Snyders, DJ
    Tamkun, MM
    Valenzuela, C
    BIOPHYSICAL JOURNAL, 1999, 76 (01) : A189 - A189
  • [10] Localization of the binding site of benzocaine on hKv1.5 channels
    Caballero, R
    Longobardo, M
    Gonzalez, T
    Valenzuela, C
    Tamargo, J
    Delpon, E
    BIOPHYSICAL JOURNAL, 2001, 80 (01) : 441A - 441A