CHARACTERIZATION OF METHOTREXATE UPTAKE BY PROTON-COUPLED FOLATE TRANSPORTER/HEME CARRIER PROTEIN 1 HETEROLOGOUSLY EXPRESSED IN HEK293 CELLS

被引:0
|
作者
Abe, Naoki [1 ]
Inoue, Katsuhisa [1 ]
Ohta, Kin-ya [1 ]
Hayashi, Yayoi [2 ]
Yuasa, Hiroaki [1 ]
机构
[1] Nagoya City Univ, Grad Sch Phamaceut Sci, Dept Biopharmaceut, Nagoya, Aichi, Japan
[2] Kinjo Gakuin Univ, Coll Pharm, Nagoya, Aichi 4638521, Japan
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
386
引用
收藏
页码:276 / 276
页数:1
相关论文
共 38 条
  • [1] Functional characterization of human proton-coupled folate transporter/heme carrier protein 1 heterologously expressed in mammalian cells as a folate transporter
    Nakai, Yasuhiro
    Inoue, Katsuhisa
    Abe, Naoki
    Hatakeyama, Mai
    Ohta, Kin-ya
    Otagiri, Masaki
    Hayashi, Yayoi
    Yuasa, Hiroaki
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2007, 322 (02): : 469 - 476
  • [2] STEREOSELECTIVITY OF THE PROTON-COUPLED FOLATE TRANSPORTER/HEME CARRIER PROTEIN 1 (PCFT/HCP1)
    Narawa, Tomoya
    Yanagisawa, Hideaki
    Tsuda, Yasuyuki
    Itoh, Tomoo
    DRUG METABOLISM REVIEWS, 2007, 39 : 164 - 164
  • [3] Purification and characterization of the creatine transporter expressed at high levels in HEK293 cells
    West, M
    Park, D
    Dodd, JR
    Kistler, J
    Christie, DL
    PROTEIN EXPRESSION AND PURIFICATION, 2005, 41 (02) : 393 - 401
  • [4] Characterization of hemichannels heterologously expressed in HEK293 cells using connexin43 linked to green fluorescent protein
    John, SA
    Wang, SY
    Weiss, JN
    CIRCULATION, 1998, 98 (17) : 11 - 12
  • [5] Site-specific contribution of proton-coupled folate transporter/haem carrier protein 1 in the intestinal absorption of methotrexate in rats
    Yokooji, Tomoharu
    Mori, Nobuhiro
    Murakami, Teruo
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 2009, 61 (07) : 911 - 918
  • [6] Haem and folate transport by proton-coupled folate transporter/haem carrier protein 1 (SLC46A1)
    Laftah, Abas H.
    Latunde-Dada, Gladys O.
    Fakih, Sarah
    Hider, Robert C.
    Simpson, Robert J.
    McKie, Andrew T.
    BRITISH JOURNAL OF NUTRITION, 2009, 101 (08) : 1150 - 1156
  • [7] Tetrahydropapaveroline and its derivatives inhibit dopamine uptake through dopamine transporter expressed in HEK293 cells
    Okada, T
    Shimada, S
    Sato, K
    Kotake, Y
    Kawai, H
    Ohta, S
    Tohyama, M
    Nishimura, T
    NEUROSCIENCE RESEARCH, 1998, 30 (01) : 87 - 90
  • [8] Activation by forskolin of the organic cation transporter ROCT1 expressed in HEK293 cells
    Hohage, I
    Lelleck, S
    Stachon, A
    Haxelmans, S
    Koepsell, H
    Schlatter, E
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1998, 358 (01) : R741 - R741
  • [9] Folate-appended cyclodextrin carrier targets ovarian cancer cells expressing the proton-coupled folate transporter
    Saito, Shinichi
    Koya, Yoshihiro
    Kajiyama, Hiroaki
    Yamashita, Mamoru
    Kikkawa, Fumitaka
    Nawa, Akihiro
    CANCER SCIENCE, 2020, 111 (05) : 1794 - 1804
  • [10] Functional Loss of the Reduced Folate Carrier Enhances the Antitumor Activities of Novel Antifolates with Selective Uptake by the Proton-Coupled Folate Transporter
    Desmoulin, Sita Kugel
    Wang, Lei
    Polin, Lisa
    White, Kathryn
    Kushner, Juiwanna
    Stout, Mark
    Hou, Zhanjun
    Cherian, Christina
    Gangjee, Aleem
    Matherly, Larry H.
    MOLECULAR PHARMACOLOGY, 2012, 82 (04) : 591 - 600