Voltage-Gated Calcium Channel Antagonists for the Central Nervous System

被引:9
作者
Barrow, James C. [1 ]
Duffy, Joseph L. [1 ]
机构
[1] Merck Res Labs, Rahway, NJ 07065 USA
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 45 | 2010年 / 45卷
关键词
PLASMA-MEMBRANE EXPRESSION; CA2+ CHANNEL; THALAMIC NEURONS; NEUROPATHIC PAIN; MICE LACKING; ABSENCE EPILEPSY; EPISODIC ATAXIA; BLOCKERS; DISCOVERY; NOMENCLATURE;
D O I
10.1016/S0065-7743(10)45001-0
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:3 / 18
页数:16
相关论文
共 50 条
[41]   Animal Venom Peptides Cause Antinociceptive Effects by Voltage-gated Calcium Channels Activity Blockage [J].
Trevisan, Gabriela ;
Oliveira, Sara Marchesan .
CURRENT NEUROPHARMACOLOGY, 2022, 20 (08) :1579-1599
[42]   The natural product argentatin C attenuates postoperative pain via inhibition of voltage-gated sodium and T-type voltage-gated calcium channels [J].
Duran, Paz ;
Loya-Lopez, Santiago ;
Ran, Dongzhi ;
Tang, Cheng ;
Calderon-Rivera, Aida ;
Gomez, Kimberly ;
Stratton, Harrison J. ;
Huang, Sun ;
Xu, Ya-ming ;
Wijeratne, E. M. Kithsiri ;
Perez-Miller, Samantha ;
Shan, Zhiming ;
Cai, Song ;
Gabrielsen, Anna T. ;
Dorame, Angie ;
Masterson, Kyleigh A. ;
Alsbiei, Omar ;
Madura, Cynthia L. ;
Luo, Guoqin ;
Moutal, Aubin ;
Streicher, John ;
Zamponi, Gerald W. ;
Gunatilaka, A. A. Leslie ;
Khanna, Rajesh .
BRITISH JOURNAL OF PHARMACOLOGY, 2023, 180 (09) :1267-1285
[43]   Spinal morphine but not ziconotide or gabapentin analgesia is affected by alternative splicing of voltage-gated calcium channel CaV2.2 pre-mRNA [J].
Jiang, Yu-Qiu ;
Andrade, Arturo ;
Lipscombe, Diane .
MOLECULAR PAIN, 2013, 9
[44]   Small-molecule CaVα1•CaVβ antagonist suppresses neuronal voltage-gated calcium-channel trafficking [J].
Chen, Xingjuan ;
Liu, Degang ;
Zhou, Donghui ;
Si, Yubing ;
Xu, David ;
Stamatkin, Christopher W. ;
Ghozayel, Mona K. ;
Ripsch, Matthew S. ;
Obukhov, Alexander G. ;
White, Fletcher A. ;
Meroueh, Samy O. .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 115 (45) :E10566-E10575
[45]   The Physiology, Pathology, and Pharmacology of Voltage-Gated Calcium Channels and Their Future Therapeutic Potential [J].
Zamponi, Gerald W. ;
Striessnig, Joerg ;
Koschak, Alexandra ;
Dolphin, Annette C. .
PHARMACOLOGICAL REVIEWS, 2015, 67 (04) :821-870
[46]   Conotoxins Targeting Neuronal Voltage-Gated Sodium Channel Subtypes: Potential Analgesics? [J].
Knapp, Oliver ;
McArthur, Jeffrey R. ;
Adams, David J. .
TOXINS, 2012, 4 (11) :1236-1260
[47]   Voltage-gated calcium channels - Moorea, April 1-7, 2007 [J].
Davies, Lucinda A. ;
Barrett, Paula Q. .
CHANNELS, 2007, 1 (02) :135-137
[48]   Voltage-Gated Calcium 2.2 Channels: Therapeutic Target for Chronic Arthritic Pain? [J].
Ashraf, Sadaf .
ARTHRITIS & RHEUMATOLOGY, 2015, 67 (06) :1416-1418
[49]   Potential roles of voltage-gated ion channel disruption in Tuberous Sclerosis Complex [J].
Egido-Betancourt, Hailey X. ;
Strowd III, Roy E. ;
Raab-Graham, Kimberly F. .
FRONTIERS IN MOLECULAR NEUROSCIENCE, 2024, 17
[50]   Conotoxins as Tools to Understand the Physiological Function of Voltage-Gated Calcium (CaV) Channels [J].
Ramirez, David ;
Gonzalez, Wendy ;
Fissore, Rafael A. ;
Carvacho, Ingrid .
MARINE DRUGS, 2017, 15 (10)