Synthesis of some new 3,4-disubstituted pyrroles and pyrazoles from E-1-(arylsulfonylethylsulfonyl)-2-arylethene

被引：0

作者：

Padmaja, A. ^{[1
]}

Syamaiah, K. ^{[1
]}

Muralikrishna, A. ^{[1
]}

Padmavathi, V. ^{[1
]}

机构：

[1] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2012年 / 51卷 / 01期

关键词：

Pyrrole; pyrazoline; pyrazole; 1,3-dipolar cycloaddition; ANTICONVULSANT ACTIVITY; DNA; ANTIBACTERIALS; POLYAMIDES; POTENT; PHASE;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The sulfonyl activated olefin. E-1-(arylsulfonylethylsulfonyl)-2-arylethene 7 has been used as a synthon to develop a new class of pyrrole and pyrazole derivatives by 1,3-dipolar cycloaddition of TosMIC and diazomethane.

引用

页码：285 / 290

页数：6

共 28 条

[1]

[Anonymous], 1992, PYRROLES 2

[2]

Black D. S. C., 1996, COMPREHENSIVE HETERO, V2, P39

[3] PYRIMIDINES .4. EXPERIMENTS ON THE SYNTHESIS OF PYRIMIDINE AND 4-6-DIMETHYLPYRIMIDINE [J].

BOARLAND, MPV ;

MCOMIE, JFW ;

TIMMS, RN .

JOURNAL OF THE CHEMICAL SOCIETY, 1952, (DEC) :4691-4695

[4] Total syntheses of ningalin A, lamellarin O, lukianol A, and permethyl storniamide A utilizing heterocyclic azadiene Diels-Alder reactions [J].

Boger, DL ;

Boyce, CW ;

Labroli, MA ;

Sehon, CA ;

Jin, Q .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1999, 121 (01) :54-62

[5] UBER NEUE 3,5-DIOXO-PYRAZOLIDINE [J].

BUCHI, J ;

AMMANN, J ;

LIEBERHERR, R ;

EICHENBERGER, E .

HELVETICA CHIMICA ACTA, 1953, 36 (01) :75-85

[6] ADDITION OF ALCOHOLS TO VINYL SULPHONES AND SULPHONAMIDES [J].

DAVIES, WG ;

HARDISTY, EW ;

NEVELL, TP ;

PETERS, RH .

JOURNAL OF THE CHEMICAL SOCIETY B-PHYSICAL ORGANIC, 1970, (05) :998-&

[7] Minor groove DNA binders as antimicrobial agents.: 1.: Pyrrole tetraamides are potent antibacterials against vancomycin resistant Enteroccoci and methicillin resistant Staphylococcus aureus [J].

Dyatkina, NB ;

Roberts, CD ;

Keicher, JD ;

Dai, YQ ;

Nadherny, JP ;

Zhang, WT ;

Schmitz, U ;

Kongpachith, A ;

Fung, K ;

Novikov, AA ;

Lou, L ;

Velligan, M ;

Khorlin, AA ;

Chen, MS .

JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (04) :805-817

[8]

FOYE WO, 1989, PRINCIPLES MED CHEM, P159

[9]

Gribble G.W., 1996, COMPREHENSIVE HETERO, V2, P207, DOI DOI 10.1016/B978-008096518-5.00043-5

[10] Design, synthesis, and biological testing of pyrazoline derivatives of combretastatin-A4 [J].

Johnson, Marlie ;

Younglove, Brent ;

Lee, Lauren ;

LeBlanc, Regan ;

Holt, Herman, Jr. ;

Hills, Patrice ;

Mackay, Hilary ;

Brown, Toni ;

Mooberry, Susan L. ;

Lee, Moses .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (21) :5897-5901

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