PharmGKB summary: isoniazid pathway, pharmacokinetics

被引:42
作者
Klein, Daniel J. [1 ,3 ]
Boukouvala, Sotiria [4 ]
McDonagh, Ellen M. [1 ]
Shuldiner, Scott R. [1 ]
Laurieri, Nicola [5 ]
Thorn, Caroline F. [1 ]
Altman, Russ B. [1 ,2 ]
Klein, Teri E. [1 ]
机构
[1] Stanford Univ, Dept Genet, Stanford, CA 94305 USA
[2] Stanford Univ, Dept Bioengn, Stanford, CA 94305 USA
[3] Univ Southern Calif, Keck Sch Med, Los Angeles, CA USA
[4] Democritus Univ Thrace, Dept Mol Biol & Genet, Alexandroupolis, Greece
[5] Univ Oxford, Dept Pharmacol, Oxford, England
关键词
anti-tuberculosis drug-induced hepatotoxicity; cytochrome P450 2E1; GSTT1; GSTM1; isoniazid; N-acetyltransferase; 2; pharmacokinetics; DRUG-INDUCED HEPATOTOXICITY; INDUCED LIVER-INJURY; N-ACETYLTRANSFERASE; S-TRANSFERASE M1; CYTOCHROME-P450; 2E1; GENOTYPE; GSTT1 GENETIC POLYMORPHISMS; SUSCEPTIBILITY RISK-FACTOR; HEPATIC BILE-ACIDS; ANTITUBERCULOSIS DRUGS; TUBERCULOSIS PATIENTS;
D O I
10.1097/FPC.0000000000000232
中图分类号
Q81 [生物工程学(生物技术)]; Q93 [微生物学];
学科分类号
071005 ; 0836 ; 090102 ; 100705 ;
摘要
[No abstract available]
引用
收藏
页码:436 / 444
页数:9
相关论文
共 114 条
[101]   Antituberculosis drug-induced hepatotoxicity: Concise up-to-date review [J].
Tostmann, Alma ;
Boeree, Martin J. ;
Aarnoutse, Rob E. ;
de lange, Wiel C. M. ;
van der Ven, Andre J. A. M. ;
Dekhuijzen, Richard .
JOURNAL OF GASTROENTEROLOGY AND HEPATOLOGY, 2008, 23 (02) :192-202
[102]  
US FDA, DRUGS FDA DAT
[103]   NOMENCLATURE FOR N-ACETYLTRANSFERASES [J].
VATSIS, KP ;
WEBER, WW ;
BELL, DA ;
DUPRET, JM ;
EVANS, DAP ;
GRANT, DM ;
HEIN, DW ;
LIN, HJ ;
MEYER, UA ;
RELLING, MV ;
SIM, E ;
SUZUKI, T ;
YAMAZOE, Y .
PHARMACOGENETICS, 1995, 5 (01) :1-17
[104]  
Vuilleumier Nicolas, 2006, Eur J Clin Pharmacol, V62, P423
[105]   NAT2 polymorphisms and susceptibility to anti-tuberculosis drug-induced liver injury: a meta-analysis [J].
Wang, P-Y. ;
Xie, S-Y. ;
Hao, Q. ;
Zhang, C. ;
Jiang, B-F. .
INTERNATIONAL JOURNAL OF TUBERCULOSIS AND LUNG DISEASE, 2012, 16 (05) :589-595
[106]   Genetic Polymorphisms of Cytochrome P450 and Glutathione S-transferase Associated with Antituberculosis Drug-induced Hepatotoxicity in Chinese Tuberculosis Patients [J].
Wang, T. ;
Yu, H. T. ;
Wang, W. ;
Pan, Y. Y. ;
He, L. X. ;
Wang, Z. Y. .
JOURNAL OF INTERNATIONAL MEDICAL RESEARCH, 2010, 38 (03) :977-986
[107]  
WEBER WW, 1985, PHARMACOL REV, V37, P25
[108]  
WHO, 2010, TREATMENT OF TUBERCULOSIS: GUIDELINES, FOURTH EDITION, P1
[109]   Localization of N-acetyltransferases NAT1 and NAT2 in human tissues [J].
Windmill, KF ;
Gaedigk, A ;
Hall, PDM ;
Samaratunga, H ;
Grant, DM ;
McManus, ME .
TOXICOLOGICAL SCIENCES, 2000, 54 (01) :19-29
[110]  
World Health Organization (WHO), 2014, Global Tuberculosis Report 2014