Transformations of 4,5,6,7-tetrahydrothieno[3,2-c]-and 1,2,3,4-tetrahydrobenzothieno[2,3-c]pyridines in reactions with alkynes activated by electron-withdrawing substituents

被引:4
作者
Voskressensky, L. G.
Borisova, T. N.
Listratova, A. V.
Sorokina, E. A.
Tolkunov, S. V.
Varlamov, A. V.
机构
[1] Peoples Friendship Univ Russia, Moscow 117198, Russia
[2] Natl Acad Sci Ukraine, LM Litvinenko Inst Physicoorgan & Coal Chem, UA-83114 Donetsk, Ukraine
基金
俄罗斯基础研究基金会;
关键词
tandem transformations; thienopyridines; benzothienopyridines; benzothieno-azocines; activated alkynes;
D O I
10.1007/s11172-007-0156-3
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The transformations of tetrahydrothieno[3,2-c]-and tetrahydrobenzothieno[2,3-c]pyridines in the reactions with acetylenedicarboxylic ester, alkyl propiolates, and acetylacetylene in alcohols were studied. Tetrahydrobenzothieno[3,2-d]azocines and 2-methoxyethyl-3-vinyl-aminoethylbenzothiophenes were synthesized.
引用
收藏
页码:1041 / 1048
页数:8
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