Synthesis and Antimicrobial Activity of N-Aryl-4-(cyano/alkoxycarbonyl)-5-(pyridin-3-yl)-1H/3H-1,2,3-triazole Derivatives

被引：6

作者：

Komsani, Jayaram Reddy ^{[1
]}

Avula, Sreenivas ^{[1
]}

Koppireddi, Satish ^{[1
]}

Koochana, Pranay Kumar ^{[2
]}

Murty, U. S. N. ^{[2
]}

Yadla, Rambabu ^{[1
]}

机构：

[1] CSIR Indian Inst Chem Technol IICT, Fluoroorgan Div, Hyderabad 500607, Andhra Pradesh, India

[2] CSIR IICT, Biol Div, Hyderabad 500607, Andhra Pradesh, India

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2015年 / 52卷 / 03期

关键词：

INTRAMOLECULAR WITTIG REACTION; SUBSTITUTED 1,2,3-TRIAZOLES; DESIGN;

D O I：

10.1002/jhet.2186

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A convenient synthesis of a new series of N-aryl-5-(pyridin-3-yl)-1H/3H-1,2,3-triazole-4-carbonitriles and alkyl N-aryl-5-(pyridin-3-yl)-1H/3H-1,2,3-triazole-4-carboxylic acid esters is reported. The newly synthesized 5-(pyridin-3-yl)-1,2,3-triazole derivatives are evaluated for their antibacterial and antifungal activity. Some of these triazole derivatives have exhibited moderate antimicrobial activity.

引用

页码：764 / 772

页数：9

共 47 条

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