Synthesis and functionalization of Indoles through palladium-catalyzed reactions

被引：1764

作者：

Cacchi, S ^{[1
]}

Fabrizi, G ^{[1
]}

机构：

[1] Univ Roma La Sapienza, Dipartimento Studi Chim & Tecnol Sostanze Biologi, I-00185 Rome, Italy

来源：

CHEMICAL REVIEWS | 2005年 / 105卷 / 07期

关键词：

D O I：

10.1021/cr040639b

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Over the past decades palladium catalysis has achieved an important place in the arsenal of organic chemists involved in the construction and functionalization of indole derivatives. Palladium-catalyzed reactions have become a very powerful tool in this area. Several areas of the palladium-catalyzed indole chemistry have been the object of an increasing number of studies, which include the development of new synthetic strategies, the optimization of reaction conditions, the utilization of solid-phase synthesis and microwave-assisted conditions, the construction of indole libraries, and the application to the synthesis of bioactive derivatives.

引用

页码：2873 / 2920

页数：48

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