Synthesis of 5-phosphoryl-substituted 1,3,4(3H)-thiadiazolones

被引：5

作者：

Kozlov, M. A. ^{[1
]}

Volkova, Y. A. ^{[1
]}

Zavarzin, I. V. ^{[1
]}

机构：

[1] Russian Acad Sci, ND Zelinsky Inst Organ Chem, 47 Leninsky Prosp, Moscow 119991, Russia

来源：

RUSSIAN CHEMICAL BULLETIN | 2019年 / 68卷 / 11期

基金：

俄罗斯科学基金会;

关键词：

5-phosphoryl-1,3,4(3H)-thiadiazol-2-ones; thiohydrazides; thiomorpholides; heterocyclization; CARBODIIMIDES; LIGANDS;

D O I：

10.1007/s11172-019-2673-2

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Reactions of various phosphorylthioformic acid morpholides with hydrazine afford phosphorylthioformhydrazides. The latter react under mild conditions with N,N '-carbonyldiimidazole to form novel 5-phosphoryl-1,3,4( 3H)-thiadiazol-2-ones.

引用

页码：2105 / 2107

页数：3

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