Acid-mediated ring expansion of 2,2-disubstituted azetidine carbamates to 6,6-disubstituted 1,3-oxazinan-2-ones

被引:0
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作者
Boddy, Alexander [1 ]
Cordier, Christopher [1 ]
Goldberg, Kristin [2 ]
Madin, Andrew [3 ]
Spivey, Alan [1 ]
Bull, James [1 ]
机构
[1] Imperial Coll London, Dept Chem, London, England
[2] AstraZeneca, Oncol, Med Chem, Cambridge, England
[3] AstraZeneca, Discovery Sci, Hit Discovery, Cambridge, England
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O6 [化学];
学科分类号
0703 ;
摘要
398-ORGN
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页数:2
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