Discovery of a novel, potent, and orally active nonpeptide antagonist of the human luteinizing hormone-releasing hormone (LHRH) receptor

被引：129
作者：
Cho, NB
Harada, M
Imaeda, T
Imada, T
Matsumoto, H
Hayase, Y
Sasaki, S
Furuya, S
Suzuki, N
Okubo, S
Ogi, K
Endo, S
Onda, H
Fujino, M
机构：
[1] Takeda Chem Ind Ltd, Div Discovery Res, Ibaraki, Osaka 3004293, Japan
[2] Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1998年 / 41卷 / 22期
关键词：
D O I：
10.1021/jm9803673
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：4190 / 4195
页数：6
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