Biphenylphosphine-palladium(II) complexes-catalyzed Friedel-Crafts Reaction for the Synthesis of α-amino and α-hydroxy indolylacetates and diindolylacetates

被引：0

作者：

Hao, J ^{[1
]}

Taktak, S ^{[1
]}

Aikawa, K ^{[1
]}

Yusa, Y ^{[1
]}

Hatano, M ^{[1
]}

Mikami, K ^{[1
]}

机构：

[1] Tokyo Inst Technol, Dept Appl Chem, Tokyo 1528552, Japan

来源：

SYNLETT | 2001年 / 09期

关键词：

biphenylphosphine; palladium complexes; Friedel-Crafts reaction; indoles;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Biphenylphosphine-palladium(II) complexes-catalyzed Friedel-Crafts reaction of N-methylindol with imino and carbonyl compounds afforded alpha -amino and alpha -hydroxy substituted indolyl-acetates and diindolylacetates in good yields.

引用

页码：1443 / 1445

页数：3

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