Preparation of tricyclic nitrogen heterocycles via tandem four-component condensation/intramolecular Diels-Alder reaction

被引：116

作者：

Paulvannan, K ^{[1
]}

机构：

[1] Affymax Res Inst, Santa Clara, CA 95051 USA

来源：

TETRAHEDRON LETTERS | 1999年 / 40卷 / 10期

关键词：

D O I：

10.1016/S0040-4039(99)00072-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Preparation of highly substituted rigid tricyclic nitrogen heterocycles via a tandem four-component condensation (4CC)/ intramolecular Diels-Alder (IMDA) reaction has been studied both in solution and solid phase. Influence of electronic and steric effects on the product formation has also been investigated. (C) 1999 Elsevier Science Ltd. All rights reserved.

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页码：1851 / 1854

页数：4

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