5-fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c][1,4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985):: An orally active arginine vasopressin antagonist with selectivity for V2 receptors

被引：140
作者：
Albright, JD [1 ]
Reich, MF
Delos Santos, EG
Dusza, JP
Sum, FW
Venkatesan, AM
Coupet, J
Chan, PS
Ru, X
Mazandarani, H
Bailey, T
机构：
[1] Wyeth Ayerst Res, Pearl River, NY 10965 USA
[2] Wyeth Ayerst Res, Princeton, NJ 08543 USA
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1998年 / 41卷 / 14期
关键词：
D O I：
10.1021/jm980179c
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：2442 / 2444
页数：3
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