5-fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c][1,4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985):: An orally active arginine vasopressin antagonist with selectivity for V2 receptors

被引：140

作者：

Albright, JD ^{[1
]}

Reich, MF

Delos Santos, EG

Dusza, JP

Sum, FW

Venkatesan, AM

Coupet, J

Chan, PS

Ru, X

Mazandarani, H

Bailey, T

机构：

[1] Wyeth Ayerst Res, Pearl River, NY 10965 USA

[2] Wyeth Ayerst Res, Princeton, NJ 08543 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1998年 / 41卷 / 14期

关键词：

D O I：

10.1021/jm980179c

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2442 / 2444

页数：3

共 33 条

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