A green development of Bernthsen 9-substituted acridine synthesis in the absence of solvent catalyzed by p-toluenesulphonic acid (p-TSA)

被引：15
作者：
Das, Subrata [1 ]
Thakur, A. J. [1 ]
机构：
[1] Cent Univ, Dept Chem Sci, Tezpur 784028, Assam, India
来源：
GREEN CHEMISTRY LETTERS AND REVIEWS | 2011年 / 4卷 / 02期
关键词：
Bernthsen; acridine; p-toluenesulphonic acid (p-TSA); microwave; ONE-ELECTRON REDUCTION; DNA; DYES; ACRIDINE-1,8-DIONE; DERIVATIVES; INHIBITORS;
D O I：
10.1080/17518253.2010.521775
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Bernthsen reaction has been carried out under microwave irradiation in the presence of p-TSA (10 mol%) as catalyst in a solventless reaction to provide 9-substituted acridines. In the present report, time economy and better yields as compared to conventional Bernthsen reaction are described.
引用
收藏
页码：131 / 135
页数：5
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