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- [1] Comparision of Dual PI-3K/mTOR Inhibitors with mTOR Inhibitors Using a Pre-Clinical Model of Acute Lymphoblastic LeukemiaBLOOD, 2010, 116 (21) : 1336 - 1336Wong, Jacky论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, Australia Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, AustraliaWelschinger, Robert论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, Australia Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, AustraliaBaraz, Rana论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, Australia Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, AustraliaWeiss, Jocelyn论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, Australia Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, AustraliaBradstock, Ken论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, AustraliaBendall, Linda J.论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Westmead Millenium Inst, Westmead Inst Canc Res, Sydney, NSW, Australia
- [2] Efficacy of dual PI-3K and mTOR inhibitors in Vitro and in Vivo in acute lymphoblastic leukemiaONCOTARGET, 2014, 5 (21) : 10460 - 10472Wong, Jacky论文数: 0 引用数: 0 h-index: 0机构: Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, Australia Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, AustraliaWelschinger, Robert论文数: 0 引用数: 0 h-index: 0机构: Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, Australia Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, AustraliaHewson, John论文数: 0 引用数: 0 h-index: 0机构: Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, Australia Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, AustraliaBradstock, Kenneth F.论文数: 0 引用数: 0 h-index: 0机构: Westmead Hosp, Dept Haematol, Westmead, NSW 2145, Australia Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, AustraliaBendall, Linda J.论文数: 0 引用数: 0 h-index: 0机构: Univ Sydney, Ctr Canc Res, Westmead Millennium Inst, Westmead, NSW 2145, Australia
- [3] Direct inhibition of mTOR may be detrimental when combining mTOR inhibitors or dual PI3 kinase/mTOR inhibitors with paclitaxelCANCER RESEARCH, 2008, 68 (09)Bhattacharya, Bhaskar论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, EnglandRichardson, Alan论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, EnglandSain, Nivedita论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, EnglandOrmerod, Michael论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, EnglandKaye, Stanley论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, EnglandWorkman, Paul论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, EnglandJackman, Ann论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, England
- [4] Activation of PI3K/Akt/mTOR Pathway and Dual Inhibitors of PI3K and mTOR in Endometrial CancerCURRENT MEDICINAL CHEMISTRY, 2014, 21 (26) : 3070 - 3080Chen, Jiezhong论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, Australia Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, AustraliaZhao, Kong-Nan论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Princess Alexandra Hosp, Sch Med, Ctr Kidney Dis Res Venom Res, Brisbane, Qld 4102, Australia Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, AustraliaLi, Rui论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, Australia Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, AustraliaShao, Renfu论文数: 0 引用数: 0 h-index: 0机构: Univ Sunshine Coast, Fac Sci Hlth Educ & Engn, GeneCol Res Ctr, Maroochydore, Qld 4556, Australia Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, AustraliaChen, Chen论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, Australia Univ Queensland, Sch Biomed Sci, St Lucia, Qld 4072, Australia
- [5] Design and synthesis of dual PI3K/mTor inhibitorsCANCER RESEARCH, 2009, 69Olivero, Alan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAHeffron, Timothy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USABerry, Leanne论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USABerry, Megan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USACastanedo, Georgette论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAChang, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USADotson, Jennafer论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAFriedman, Lori论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAGoldsmith, Richard论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USALesnick, John论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USALewis, Cristina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAMathieu, Simon论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USANonomiya, Jim论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAPang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAPeterson, David论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAPrior, Wei Wei论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USASampath, Deepak论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USASutherlin, Daniel论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USATsui, Vickie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAUltsch, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAWang, Shumei论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAWiesmann, Christian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAWong, Susan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAZhu, Bing-Yan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAChuckowree, Irina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAFolkes, Adrian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USAShuttleworth, Steve论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA
- [6] Dual PI3K and mTOR Inhibition in Waldenstrom MacroglobulinemiaCLINICAL LYMPHOMA & MYELOMA, 2009, 9 : S144 - S145Husu, E. N.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USARoccaro, A. M.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAAnderson, K. C.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAGhobrial, I. M.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USALeleu, X.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USASacco, A.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAMelhem, M. R.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAAzab, A. K.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAJia, X.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USANgo, H. T.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAAzab, F.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USARunnels, J.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USAQuang, P.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA
- [7] Inhibition of mTOR, but not PI3K, is required for the anti-tumor efficacy in breast cancer of dual PI3K/mTOR inhibitors given in combination with MEK inhibitorsCANCER RESEARCH, 2015, 75Smith, Aleisha M.论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USAXiong, Jessie论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USAHunter, Lucas论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USAJordan, Jamie论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USAClark, Kelly论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USADarr, David B.论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USANorman, Sharpless论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USAPerou, Charles M.论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USAKim, William Y.论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA UNC Lineberger Comp Ctr Canc, Chapel Hill, NC USA
- [8] Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 211Alvarez, Rosa M.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainBelen Garcia, Ana论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainRiesco-Fagundo, Concepcion论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainMartin, Jose, I论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain GSK, Med Chem, Dis Developing World, C Severo Ochoa 2,Sci Business Technol Pk, E-28760 Tres Cantos, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainVarela, Carmen论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainRodriguez Hergueta, Antonio论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Ctr Invest Lilly SA, Avda Ind 30, E-28108 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainGonzalez Cantalapiedra, Esther论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainOyarzabal, Julen论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Univ Navarra, CIMA, Ctr Appl Med Res, Mol Therapeut Program,Small Mol Discovery Platfor, Avda Pio XII 55, Pamplona 31008, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainDi Geronimo, Bruno论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainLorenzo, Milagros论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainIsabel Albarran, M.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainCebria, Antonio论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain GSK, Dis Developing World, Pharmacol Unit, C Severo Ochoa 2,Sci Business Technol Pk, E-28760 Tres Cantos, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainCebrian, David论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainMartinez-Gonzalez, Sonia论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainBlanco-Aparicio, Carmen论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, SpainPastor, Joaquin论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain Spanish Natl Canc Res Ctr CNIO, Expt Therapeut Programme, C Melchor Fernandez Almagro 3, E-28029 Madrid, Spain
- [9] Dual Inhibitors of PI3K/mTOR or mTOR-Selective Inhibitors: Which Way Shall We Go?CURRENT MEDICINAL CHEMISTRY, 2011, 18 (36) : 5528 - 5544Sabbah, D. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Nebraska Med Ctr, Coll Pharm, Omaha, NE 68198 USA Univ Nebraska, Dept Chem, Omaha, NE 68182 USABrattain, M. G.论文数: 0 引用数: 0 h-index: 0机构: Univ Nebraska Med Ctr, Eppley Canc Inst, Omaha, NE 68198 USA Univ Nebraska, Dept Chem, Omaha, NE 68182 USAZhong, H.论文数: 0 引用数: 0 h-index: 0机构: Univ Nebraska, Dept Chem, Omaha, NE 68182 USA Univ Nebraska, Dept Chem, Omaha, NE 68182 USA
- [10] Dueling for dual inhibition: Means to enhance effectiveness of PI3K/Akt/mTOR inhibitors in AMLBLOOD REVIEWS, 2018, 32 (03) : 235 - 248Herschbein, Lauren论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Dept Med, James P Wilmot Canc Inst, Rochester, NY 14627 USA Univ Rochester, Dept Med, James P Wilmot Canc Inst, Rochester, NY 14627 USALiesveld, Jane L.论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Dept Med, James P Wilmot Canc Inst, Rochester, NY 14627 USA Univ Rochester, Dept Med, James P Wilmot Canc Inst, Rochester, NY 14627 USA