共 153 条
Multimodal Role of PACAP in Glioblastoma
被引:17
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Pittala, Valeria
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Univ Catania, Dept Drug & Hlth Sci, I-95125 Catania, Italy Univ Catania, Dept Drug & Hlth Sci, I-95125 Catania, Italy

Reglodi, Dora
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机构:
Univ Pecs, Med Sch, Dept Anat, MTA PTE PACAP Res Grp, H-7624 Pecs, Hungary Univ Catania, Dept Drug & Hlth Sci, I-95125 Catania, Italy

D'Agata, Velia
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Univ Catania, Sect Anat Histol & Movement Sci, Dept Biomed & Biotechnol Sci, I-95100 Catania, Italy Univ Catania, Dept Drug & Hlth Sci, I-95125 Catania, Italy
机构:
[1] Univ Catania, Dept Drug & Hlth Sci, I-95125 Catania, Italy
[2] Univ Catania, Sect Anat Histol & Movement Sci, Dept Biomed & Biotechnol Sci, I-95100 Catania, Italy
[3] Univ Pecs, Med Sch, Dept Anat, MTA PTE PACAP Res Grp, H-7624 Pecs, Hungary
关键词:
glioblastoma multiforme;
tumoral microenvironment;
hypoxia;
PACAP;
CYCLASE-ACTIVATING POLYPEPTIDE;
VASOACTIVE-INTESTINAL-PEPTIDE;
GROWTH-FACTOR RECEPTOR;
4 SPLICE VARIANTS;
STEM-LIKE CELLS;
ADENYLATE-CYCLASE;
EXTRACELLULAR DOMAIN;
SIGNAL-TRANSDUCTION;
SURVIVAL BENEFIT;
NERVOUS-SYSTEM;
D O I:
10.3390/brainsci11080994
中图分类号:
Q189 [神经科学];
学科分类号:
071006 ;
摘要:
Glioblastoma multiforme (GBM) is the deadliest form of brain tumors. To date, the GBM therapeutical approach consists of surgery, radiation-therapy and chemotherapy combined with molecules improving cancer responsiveness to treatments. In this review, we will present a brief overview of the GBM classification and pathogenesis, as well as the therapeutic approach currently used. Then, we will focus on the modulatory role exerted by pituitary adenylate cyclase-activating peptide, known as PACAP, on GBM malignancy. Specifically, we will describe PACAP ability to interfere with GBM cell proliferation, as well as the tumoral microenvironment. Considering its anti-oncogenic role in GBM, synthesis of PACAP agonist molecules may open new perspectives for combined therapy to existing gold standard treatment.
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