CS-917, a fructose 1,6-bisphosphatase inhibitor, reduces plasma glucose by suppressing hepatic glucose production, whereas metformin stimulates gastrointestinal glucose uptake

被引:0
作者
Okuno, A. [1 ]
Tanaka, J. [1 ]
Takahashi, K. [1 ]
Ogawa, J. [1 ]
Hagisawa, Y. [1 ]
Kanda, S. [1 ]
Yoshida, T. [1 ]
机构
[1] Daiichi Sankyo Co Ltd, Biol Res Labs 2, Tokyo, Japan
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D O I
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中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
0218
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页码:S95 / S95
页数:1
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[31]   The Ancient Drug Salicylate Indirectly Targets Fructose-1,6-Bisphosphatase to Suppress Liver Glucose Production in Diet-Induced Obese Mice [J].
Nisr, Raid B. ;
Atrih, Abdelmadjid ;
Lara, Erika J. Gutierrez ;
Lamont, Douglas ;
Luda, Katarzyna M. ;
Mccrimmon, Rory J. ;
Sakamoto, Kei ;
Rena, Graham ;
McNeilly, Alison D. .
ACTA PHYSIOLOGICA, 2025, 241 (06)
[32]   INDUCTION OF FRUCTOSE 1,6-BISPHOSPHATASE AND GLUCOSE 6-PHOSPHATASE BY DIBUTYRYL CYCLIC ADENOSINE-MONOPHOSPHATE IN FETAL MOUSE-LIVER [J].
TASHIMA, Y ;
MIZUNUMA, H ;
SHIMA, H ;
KOBAYASHI, R ;
TANAKA, S ;
MAEDA, N ;
KUMEGAWA, M .
JOURNAL OF BIOCHEMISTRY, 1984, 96 (03) :805-813
[33]   EFFECT OF ADRENERGIC AGONISTS AND ANTAGONISTS ON ALANINE AMINO TRANSFERASE, FRUCTOSE-1 - 6-BISPHOSPHATASE AND GLUCOSE-PRODUCTION IN HEPATOCYTES [J].
BEGUM, NA ;
DATTA, AG .
MOLECULAR AND CELLULAR BIOCHEMISTRY, 1992, 113 (02) :93-103
[34]   A potential role for muscle in glucose homeostasis: in vivo kinetic studies in glycogen storage disease type 1a and fructose-1,6-bisphosphatase deficiency [J].
Huidekoper, Hidde H. ;
Visser, Gepke ;
Ackermans, Mariette T. ;
Sauerwein, Hans P. ;
Wijburg, Frits A. .
JOURNAL OF INHERITED METABOLIC DISEASE, 2010, 33 (01) :25-31
[35]   Dehydroepiandrosterone suppresses the elevated hepatic glucose-6-phosphatase and fructose-1,6-bisphosphatase activities in C57BL/Ksj-db/db mice -: Comparison with troglitazone [J].
Aoki, K ;
Saito, T ;
Satoh, S ;
Mukasa, K ;
Kaneshiro, M ;
Kawasaki, S ;
Okamura, A ;
Sekihara, H .
DIABETES, 1999, 48 (08) :1579-1585
[36]   Pronounced and rapid glucose lowering with the fructose-1,6-bisphosphatase (FBPase) inhibitor MB07803 in poorly controlled type 2 diabetes mellitus (T2DM) subjects [J].
Gumbiner, B. ;
Watling, S. ;
Milad, M. ;
Stern, T. ;
Longcore, A. ;
Le, T. ;
Fereshetian, A. ;
Foyt, H. ;
Erion, M. .
DIABETOLOGIA, 2009, 52 :S343-S343
[37]   Molecular characterization of fructose-1,6-bisphosphatase 1b in blunt snout bream Megalobrama amblycephala and the transcriptional response to glucose loading after the adaptation to high-carbohydrate diets [J].
Li, Xiang-Fei ;
Xu, Chao ;
Jiang, Guang-Zhen ;
Zhang, Ding-Dong ;
Liu, Wen-Bin .
FISH PHYSIOLOGY AND BIOCHEMISTRY, 2017, 43 (05) :1337-1349
[38]   Molecular characterization of fructose-1,6-bisphosphatase 1b in blunt snout bream Megalobrama amblycephala and the transcriptional response to glucose loading after the adaptation to high-carbohydrate diets [J].
Xiang-Fei Li ;
Chao Xu ;
Guang-Zhen Jiang ;
Ding-Dong Zhang ;
Wen-Bin Liu .
Fish Physiology and Biochemistry, 2017, 43 :1337-1349
[39]   Regulation of hepatic glucose production and AMPK by AICAR but not by metformin depends on drug uptake through the equilibrative nucleoside transporter 1 (ENT1) [J].
Logie, Lisa ;
Lees, Zoe ;
Allwood, J. William ;
McDougall, Gordon ;
Beall, Craig ;
Rena, Graham .
DIABETES OBESITY & METABOLISM, 2018, 20 (12) :2748-2758
[40]   HYPOGLYCEMIC ACTIVITY OF COCCINIA-INDICA AND MOMORDICA-CHARANTIA IN DIABETIC RATS - DEPRESSION OF THE HEPATIC GLUCONEOGENIC ENZYMES GLUCOSE-6-PHOSPHATASE AND FRUCTOSE-1,6-BISPHOSPHATASE AND ELEVATION OF BOTH LIVER AND RED-CELL SHUNT ENZYME GLUCOSE-6-PHOSPHATE-DEHYDROGENASE [J].
SHIBIB, BA ;
KHAN, LA ;
RAHMAN, R .
BIOCHEMICAL JOURNAL, 1993, 292 :267-270