Synthesis of New Pyrazolopyrimidinedithiones and Pyrazolopyrimidinephosphines from Aminocyanopyrazoles

被引:10
作者
Allouche, Fatma [1 ]
Chabchoub, Fahker [1 ]
Salem, Mansour [1 ]
Kirsch, Gilbert [2 ]
机构
[1] Fac Sci Sfax, Lab Chim Appl Heterocycles Corps Gras & Polymeres, Sfax 3018, Tunisia
[2] CNRS, Inst Jean Barriol, Lab Ingn Mol & Biochim Pharmacol, Metz, France
关键词
Pyrazole; pyrazolopyrimidinedithione; pyrazolopyrimidinephosphine; DERIVATIVES; PYRAZOLE; ACIDS;
D O I
10.1080/00397911.2010.486516
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[image omitted] A general, high-yielding synthetic protocol for the expedited synthesis of functionalized pyrazolopyrimidine dithione 2 and pyrazolodiazaphosphininethione 3 from amino-cyano pyrazole 1 precursors is presented.
引用
收藏
页码:1500 / 1507
页数:8
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