共 66 条
Inflammation-Responsive Drug-Loaded Hydrogels with Sequential Hemostasis, Antibacterial, and Anti-Inflammatory Behavior for Chronically Infected Diabetic Wound Treatment
被引:286
作者:

Wang, Yu
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Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Wu, Ye
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Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Long, Linyu
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Sichuan Univ, Natl Engn Res Ctr Biomat, Chengdu 610064, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Yang, Li
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Sichuan Univ, Natl Engn Res Ctr Biomat, Chengdu 610064, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Fu, Daihua
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Sichuan Univ, Natl Engn Res Ctr Biomat, Chengdu 610064, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Hu, Cheng
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Sichuan Univ, Natl Engn Res Ctr Biomat, Chengdu 610064, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Kong, Qingquan
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Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China
Sichuan Univ, Med X Ctr Mat, Chengdu 610064, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China

Wang, Yunbing
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Sichuan Univ, Natl Engn Res Ctr Biomat, Chengdu 610064, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China
机构:
[1] Sichuan Univ, West China Hosp, Dept Orthoped, Orthoped Res Inst, Chengdu 610041, Sichuan, Peoples R China
[2] Sichuan Univ, Natl Engn Res Ctr Biomat, Chengdu 610064, Sichuan, Peoples R China
[3] Sichuan Univ, Med X Ctr Mat, Chengdu 610064, Sichuan, Peoples R China
关键词:
inflammation-responsive;
hemostasis;
antibacterial hybrid;
drug-loaded micelles;
wound healing;
INJECTABLE HYDROGELS;
IN-VITRO;
NANOPARTICLES;
GELATIN;
NANOCLUSTERS;
MECHANISMS;
MICELLES;
ALGINATE;
DELIVERY;
POLYMER;
D O I:
10.1021/acsami.1c09889
中图分类号:
TB3 [工程材料学];
学科分类号:
0805 ;
080502 ;
摘要:
Stimuli-responsive hydrogels possess unique advantages in drug delivery due to their variable performance and status based on the external environment. In the present study, a dual-responsive (pH and reactive oxygen species (ROS)) hydrogel was prepared to realize drug release properties under inflammatory stimulation. By grafting 3-carboxy-phenylboronic acid to the gelatin molecular backbone and cross-linking with poly(vinyl alcohol), we successfully synthesized the inflammation-responsive drug-loaded hydrogels after encapsulation with vancomycin-conjugated silver nanoclusters (VAN-AgNCs) and pH-sensitive micelles loaded with nimesulide (NIM). This novel design not only retained the dynamic functions of hydrogels, such as injectability, self-healing, and remodeling, but also realized sequential and on-demand drug delivery at diabetic-infected wound sites. In this work, we found that the hydrogel exhibited excellent biocompatibility and hemostasis properties owing to the enhanced cell-adhesive property of the gelatin component. The significant antibacterial and anti-inflammatory effect of the hydrogel was demonstrated in an in vitro experiment. Moreover, in the in vivo experiment, the hydrogel was found to play a role in promoting infected wound healing through sequential hemostasis and anti-bacterial and anti-inflammatory processes. Collectively, this inflammation-responsive hydrogel design containing VAN-AgNCs and NIM-loaded micelles has great potential in the application of chronically infected diabetic wound treatment, as well as in other inflammatory diseases.
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收藏
页码:33584 / 33599
页数:16
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Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China

Guo, Qianqian
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Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China

Zhao, Yu
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Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China

Zhang, Peng
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Univ Washington, Dept Chem Engn, Seattle, WA 98195 USA Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China

Zhang, Tianqi
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Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China

Zhang, Xinge
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Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China

Li, Chaoxing
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Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China Nankai Univ, Inst Polymer Chem, Minist Educ, Key Lab Funct Polymer Mat, Tianjin 300071, Peoples R China
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Dalton, B. R.
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Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Rajakumar, I
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Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Langevin, A.
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Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Ondro, C.
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Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Sabuda, D.
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Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Griener, T. P.
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Univ Calgary, Dept Pathol & Lab Med, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Dersch-Mills, D.
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Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada

Rennert-May, E.
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Univ Calgary, Dept Med, Sect Infect Dis, Calgary, AB, Canada Alberta Hlth Serv, Pharm Serv, Calgary, AB, Canada