Synthesis of Pyrazole Compounds by Using Sonication Method

被引：2

作者：

Kumdale, Prashant Ganpatrao ^{[1
]}

Shitole, Nana Vikram ^{[2
]}

机构：

[1] Shivneri Coll, Dept Chem, Shirur Anantpal, MS, India

[2] Shri Shivaji Coll Parbhani MS, Dept Chem, Parbhani 431401, MS, India

来源：

ORIENTAL JOURNAL OF CHEMISTRY | 2022年 / 38卷 / 01期

关键词：

Substituted; 1H-pyrazoles; Sonication; Hydrazine hydrate; Cyclo condensation; ONE-POT SYNTHESIS; BIOLOGICAL EVALUATION; 1,3-DIPOLAR CYCLOADDITION; ASSISTED SYNTHESIS; DERIVATIVES; INHIBITORS; HYDRAZINES; EFFICIENT; SELECTIVITY; SILDENAFIL;

D O I：

10.13005/ojc/380125

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

A simple method for the synthesis of pyrazoles derivatives carried out by cyclization of cyanide with hydrazine hydrate by using sonication method. All the prepared compounds were characterized by H-1, C-13 NMR and IR Spectroscopy.

引用

页码：198 / 203

页数：6

共 52 条

[1] Synthesis and structure-activity relationship of a new series of potent AT(1) selective angiotensin II receptor antagonists: 5-(biphenyl-4-ylmethyl)pyrazoles [J].

Almansa, C ;

Gomez, LA ;

Cavalcanti, FL ;

deArriba, AF ;

GarciaRafanell, J ;

Forn, J .

JOURNAL OF MEDICINAL CHEMISTRY, 1997, 40 (04) :547-558

[2]

Asirvatham S, 2021, Journal of Chemical Reviews, V3, P247, DOI [10.22034/jcr.2021.295839.1123, 10.22034/jcr.2021.295839.1123, 10.22034/JCR.2021.295839.1123, DOI 10.22034/JCR.2021.295839.1123]

[3] Synthesis of Substituted Pyrazoles via Tandem Cross-Coupling/Electrocyclization of Enol Triflates and Diazoacetates [J].

Babinski, David J. ;

Aguilar, Hector R. ;

Still, Raymond ;

Frantz, Doug E. .

JOURNAL OF ORGANIC CHEMISTRY, 2011, 76 (15) :5915-5923

[4] 4-3(5)-PYRAZOLYLPYRIDINIUM SALTS - A NEW CLASS OF HYPOGLYCEMIC AGENTS [J].

BAUER, VJ ;

DALALIAN, HP ;

FANSHAWE, WJ ;

SAFIR, SR ;

TOCUS, EC ;

BOSHART, CR .

JOURNAL OF MEDICINAL CHEMISTRY, 1968, 11 (05) :981-&

[5]

Bukhari SNA, 2012, MINI-REV MED CHEM, V12, P1394

[6] Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones [J].

Castagnolo, Daniele ;

Manetti, Fabrizio ;

Radi, Marco ;

Bechi, Beatrice ;

Pagano, Mafalda ;

De Logu, Alessandro ;

Meleddu, Rita ;

Saddi, Manuela ;

Botta, Maurizio .

BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 17 (15) :5716-5721

[7] The chemical development of the commercial route to sildenafil: A case history [J].

Dale, DJ ;

Dunn, PJ ;

Golightly, C ;

Hughes, ML ;

Levett, PC ;

Pearce, AK ;

Searle, PM ;

Ward, G ;

Wood, AS .

ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2000, 4 (01) :17-22

[8]

Dang T. T., 2011, SYNLETT, V26, P33

[9] PYRAZOLODIAZEPINES .3. 4-ARYL-1,6,7,8-TETRAHYDRO-1,3-DIALKYLPYRAZOLO[3,4-E][1,4]DIAZEPINES AS ANTI-DEPRESSANT AGENTS [J].

DEWALD, HA ;

LOBBESTAEL, S ;

POSCHEL, BPH .

JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (08) :982-987

[10] Discovery of a potent and selective series of pyrazole bacterial methionyl-tRNA synthetase inhibitors [J].

Finn, J ;

Mattia, K ;

Morytko, M ;

Ram, S ;

Yang, YF ;

Wu, XM ;

Mak, E ;

Gallant, P ;

Keith, D .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2003, 13 (13) :2231-2234

← 1 2 3 4 5 6 →