Amcenestrant in combination with CDK4/6 inhibitor palbociclib demonstrates synergistic anti-tumor activity in ER plus endocrine-resistant breast cancer xenograft models

被引:1
作者
Shomali, Maysoun
Guo, Zhuyan
Cheng, Jane
Sullivan, Amy
El-Ahmad, Youssef
Sun, Fangxian
Sidhu, Sukhvinder
Lee, Joon Sang
Cai, Hui
Pollard, Jack
Debussche, Laurent
Soria, Chris
Bouaboula, Monsif
机构
关键词
D O I
10.1158/1538-7445.SABCS21-P4-02-08
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
P4-02-08
引用
收藏
页数:2
相关论文
共 50 条
[21]   CDK4/6 inhibitor-resistant ER plus breast cancer cell lines are hypersensitive to TTK inhibition [J].
Bretones, Isabel Soria ;
Thu, Kelsie L. ;
Silvester, Jennifer ;
Kiarash, Reza ;
Fletcher, Graham C. ;
Cruickshank, Jennifer ;
Bray, Mark R. ;
Mak, Tak W. ;
Cescon, David W. .
CANCER RESEARCH, 2020, 80 (04)
[22]   Synergistic anti-tumor activity of CDK4/6 inhibitor combined with paclitaxel in NSCLC cells harboring mutant KRAS [J].
Zhang, Xiang-Hua ;
Shin, Jung-Young ;
Kim, Jeong-Oh ;
Oh, Ji-Eun ;
Chae, Hiun Suk ;
Kang, Jin-Hyoung .
CANCER RESEARCH, 2012, 72
[23]   Glucose Metabolic Reprogramming of ER+ Breast Cancer in Acquired Resistance to the CDK4/6 Inhibitor Palbociclib [J].
Lorito, Nicla ;
Bacci, Marina ;
Smiriglia, Alfredo ;
Mannelli, Michele ;
Parri, Matteo ;
Comito, Giuseppina ;
Ippolito, Luigi ;
Giannoni, Elisa ;
Bonechi, Martina ;
Benelli, Matteo ;
Migliaccio, Ilenia ;
Malorni, Luca ;
Chiarugi, Paola ;
Morandi, Andrea .
CELLS, 2020, 9 (03)
[24]   Anti-cell growth and anti-cancer stem cell activity of the CDK4/6 inhibitor palbociclib in breast cancer cells [J].
Kishino, Emi ;
Ogata, Ryohei ;
Saitoh, Wataru ;
Koike, Yoshikazu ;
Ohta, Yusuke ;
Kanomata, Naoki ;
Kurebayashi, Junichi .
BREAST CANCER, 2020, 27 (03) :415-425
[25]   Anti-cell growth and anti-cancer stem cell activity of the CDK4/6 inhibitor palbociclib in breast cancer cells [J].
Emi Kishino ;
Ryohei Ogata ;
Wataru Saitoh ;
Yoshikazu Koike ;
Yusuke Ohta ;
Naoki Kanomata ;
Junichi Kurebayashi .
Breast Cancer, 2020, 27 :415-425
[26]   AP-1 as a potential mediator of resistance to the cyclin-dependent kinase (CDK) 4/6-inhibitor palbociclib in ER-positive endocrine-resistant breast cancer [J].
De Angelis, Carmine ;
Nardone, Agostina ;
Cataldo, Maria Letizia ;
Veeraraghavan, Jamunarani ;
Fu, Xiaoyong ;
Giuliano, Mario ;
Malorni, Luca ;
Jeselsohn, Rinath ;
Osborne, Kent C. ;
Schiff, Rachel .
CANCER RESEARCH, 2018, 78 (04)
[27]   Co-targeting CDK4/6 and AKT with endocrine therapy prevents progression in CDK4/6 inhibitor and endocrine therapy-resistant breast cancer [J].
Alves, Carla L. ;
Ehmsen, Sidse ;
Terp, Mikkel G. ;
Portman, Neil ;
Tuttolomondo, Martina ;
Gammelgaard, Odd L. ;
Hundebol, Monique F. ;
Kaminska, Kamila ;
Johansen, Lene E. ;
Bak, Martin ;
Honeth, Gabriella ;
Bosch, Ana ;
Lim, Elgene ;
Ditzel, Henrik J. .
NATURE COMMUNICATIONS, 2021, 12 (01)
[28]   Longitudinal, multimodal profiling of metastatic ER plus breast cancer on CDK4/6 inhibitor therapy [J].
Creason, Allison L. ;
Egger, Julian ;
Watson, Cameron ;
Sivagnanam, Shamilene ;
Lin, Jia-Ren ;
Chin, Koei ;
Sorger, Peter K. ;
Coussens, Lisa M. ;
Mitri, Zahi I. ;
Gray, Joe W. ;
Mills, Gordon B. ;
Goecks, Jeremy .
CANCER RESEARCH, 2023, 83 (07)
[29]   G1T48, an oral selective estrogen receptor degrader, and the CDK4/6 inhibitor lerociclib inhibit tumor growth in animal models of endocrine-resistant breast cancer [J].
Andreano, Kaitlyn J. ;
Wardell, Suzanne E. ;
Baker, Jennifer G. ;
Desautels, Taylor K. ;
Baldi, Robert ;
Chao, Christina A. ;
Heetderks, Kendall A. ;
Bae, Yeeun ;
Xiong, Rui ;
Tonetti, Debra A. ;
Gutgesell, Lauren M. ;
Zhao, Jiong ;
Sorrentino, Jessica A. ;
Thompson, Delita A. ;
Bisi, John E. ;
Strum, Jay C. ;
Thatcher, Gregory R. J. ;
Norris, John D. .
BREAST CANCER RESEARCH AND TREATMENT, 2020, 180 (03) :635-646
[30]   G1T48, an oral selective estrogen receptor degrader, and the CDK4/6 inhibitor lerociclib inhibit tumor growth in animal models of endocrine-resistant breast cancer [J].
Kaitlyn J. Andreano ;
Suzanne E. Wardell ;
Jennifer G. Baker ;
Taylor K. Desautels ;
Robert Baldi ;
Christina A. Chao ;
Kendall A. Heetderks ;
Yeeun Bae ;
Rui Xiong ;
Debra A. Tonetti ;
Lauren M. Gutgesell ;
Jiong Zhao ;
Jessica A. Sorrentino ;
Delita A. Thompson ;
John E. Bisi ;
Jay C. Strum ;
Gregory R. J. Thatcher ;
John D. Norris .
Breast Cancer Research and Treatment, 2020, 180 :635-646