Sterically geared tris-thioureas; transmembrane chloride transporters with unusual activity and accessibility

被引:37
作者
Valkenier, Hennie [1 ]
Dias, Christopher M. [1 ]
Goff, Kathryn L. Porter [1 ]
Jurcek, Ondrej [2 ]
Puttreddy, Rakesh [2 ]
Rissanen, Kari [2 ]
Davis, Anthony P. [1 ]
机构
[1] Univ Bristol, Sch Chem, Bristol BS8 1TS, Avon, England
[2] Univ Jyvaskyla, Dept Chem, Nanoscience Ctr, FI-40014 Jyvaskyla, Finland
基金
英国工程与自然科学研究理事会;
关键词
ANION TRANSPORTERS; BINDING CONSTANTS; RECOGNITION; ANIONOPHORES; AFFINITIES; RECEPTORS; SENSOR; ASSAY;
D O I
10.1039/c5cc05737j
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Tris-N-arylthioureas derived in one step from 1,3,5-tris(aminomethyl)-2,4,6-triethylbenzene are remarkably effective anion carriers. With optimised aryl substituents their activities come close to the best currently known, suggesting that they might find use as readily available standards in anion transport research.
引用
收藏
页码:14235 / 14238
页数:4
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