MECHANISM-BASED INHIBITORS OF GLYCOSIDASES: DESIGN AND APPLICATIONS

被引：28

作者：

Kallemeijn, Wouter W. ^{[1
]}

Witte, Martin D. ^{[2
]}

Wennekes, Tom ^{[3
]}

Aerts, Johannes M. F. G. ^{[1
]}

机构：

[1] Univ Amsterdam, Acad Med Ctr, Dept Med Biochem, NL-1105 AZ Amsterdam, Netherlands

[2] Univ Groningen, Dept Bioorgan Chem, Stratingh Inst Chem, Groningen, Netherlands

[3] Wageningen Univ, Dept Synthet Organ Chem, NL-6700 AP Wageningen, Netherlands

来源：

ADVANCES IN CARBOHYDRATE CHEMISTRY AND BIOCHEMISTRY, VOL 71 | 2014年 / 71卷

关键词：

ACID-BETA-GLUCOSIDASE; GLYCOSYL-ENZYME INTERMEDIATE; ACTIVE-SITE NUCLEOPHILE; ACTIVITY-BASED PROBES; GLUCOCEREBROSIDE-CLEAVING ENZYME; LACTASE-PHLORHIZIN HYDROLASE; SUBSTRATE-ASSISTED CATALYSIS; SUCRASE-ISOMALTASE COMPLEX; PROTEIN-PROFILING PROBES; X-RAY CRYSTALLOGRAPHY;

D O I：

10.1016/B978-0-12-800128-8.00004-2

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：297 / 338

页数：42

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