Synthesis of Poly-Substituted Quinolines via Friedlander Hetero-Annulation Reaction Using Silica-Supported P2O5 under Solvent-Free Conditions

被引：0

作者：

Hasaninejad, Alireza ^{[1
]}

Zare, Abdolkarim ^{[2
]}

Zolfigol, Mohammad Ali ^{[3
]}

Abdeshah, Marzieh ^{[1
]}

Ghaderi, Arash ^{[1
]}

Nami-Ana, Fatemeh ^{[1
]}

机构：

[1] Persian Gulf Univ, Fac Sci, Dept Chem, Bushehr, Iran

[2] PNU, Dept Chem, Tehran, Iran

[3] Bu Ali Sina Univ, Fac Chem, Hamadan, Iran

来源：

IRANIAN JOURNAL OF CHEMISTRY & CHEMICAL ENGINEERING-INTERNATIONAL ENGLISH EDITION | 2011年 / 30卷 / 01期

关键词：

Quinoline; Friedlander hetero-annulation; P2O5/SiO2; Solvent-free; Green chemistry; ONE-POT SYNTHESIS; SULFURIC-ACID; CARBONYL-COMPOUNDS; EFFICIENT REAGENT; HIGHLY EFFICIENT; FUNCTIONALIZED QUINOLINES; MICROWAVE IRRADIATION; CONJUGATED POLYMERS; AMINOARYL KETONES; SULFONIC-ACID;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A highly efficient, simple and green solvent-free protocol for the preparation of poly-substituted quinolines via Friedlander hetero-annulation reaction between 2-aminoaryl ketones and carbonyl compounds in the presence of silica-supported P2O5(P2O5/SiO2) is described. In this method, the title compounds are obtained in high to excellent yields and in short reaction times. [GRAPHICS]

引用

页码：73 / 81

页数：9

共 64 条

[1] NEW CONJUGATED POLYANTHRAZOLINES CONTAINING THIOPHENE MOIETIES IN THE MAIN CHAIN [J].

AGRAWAL, AK ;

JENEKHE, SA .

MACROMOLECULES, 1991, 24 (25) :6806-6808

[2] Selective Oxidation of Benzylic and Allylic Alcohols with NaOCl/Silica Gel System [J].

Alinezhad, H. ;

Tajbakhsh, M. ;

Soleimani, R. .

JOURNAL OF THE IRANIAN CHEMICAL SOCIETY, 2009, 6 (02) :288-292

[3] A new green approach to the Friedlander synthesis of quinolines [J].

Arcadi, A ;

Chiarini, M ;

Di Giuseppe, S ;

Marinelli, F .

SYNLETT, 2003, (02) :203-206

[4] New vistas in quinoline synthesis [J].

Atechian, Sarkis ;

Nock, Nadine ;

Norcross, Roger D. ;

Ratni, Hassen ;

Thomas, Andrew W. ;

Verron, Julien ;

Masciadri, Raffaello .

TETRAHEDRON, 2007, 63 (13) :2811-2823

[5]

Badri, 2007, SYNTHETIC COMMUN, V37, P631

[6] Identification of xanthurenic acid as the putative inducer of malaria development in the mosquito [J].

Billker, O ;

Lindo, V ;

Panico, M ;

Etienne, AE ;

Paxton, T ;

Dell, A ;

Rogers, M ;

Sinden, RE ;

Morris, HR .

NATURE, 1998, 392 (6673) :289-292

[7] An efficient, high yielding protocol for the synthesis of functionalized quinolines via the tandem addition/annulation reaction of o-aminoaryl ketones with α-methylene ketones [J].

Bose, DS ;

Kumar, RK .

TETRAHEDRON LETTERS, 2006, 47 (05) :813-816

[8]

CHENG CC, 1982, ORG REACTIONS, V28, P37

[9]

CHO CS, 2000, J CHEM SOC CHEM COMM, V1885

[10]

Clark J.H., 2000, RSC CLEAN TECHNOL MO

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