PHASE TRANSFER-CATALYZED, ONE-POT SYNTHESIS OF SOME NOVEL N-PYRIMIDINYL-N′-NICOTINYL THIOUREA DERIVATIVES

被引:119
作者
Liu, Xing-Hai [1 ]
Tan, Cheng-Xia [1 ]
Weng, Jian-Quan [1 ]
机构
[1] Zhejiang Univ Technol, Coll Chem Engn & Mat Sci, Hangzhou 310014, Zhejiang, Peoples R China
基金
中国国家自然科学基金;
关键词
Acyl thiourea; fungicidal activity; one-pot synthesis; phase transfer catalysis;
D O I
10.1080/10426507.2010.508059
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
A new series of acyl thiourea derivatives were synthesized in one-pot using PEG-600 as the phase transfer catalyst (PTC). The structures of title compounds were characterized by H-1 NMR, IR, MS, and elemental analysis. In addition, the fungicidal activity of the acyl thiourea derivatives were tested, which showed that most of them exhibit moderate activity.
引用
收藏
页码:552 / 557
页数:6
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