Discovery of TAK-137 and TAK-653, clinical candidates of α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid receptor potentiators with reduced agonistic activities

被引:0
|
作者
Nakamura, Shinji [1 ]
Toyofuku, Masashi [1 ]
Honda, Eiji [1 ]
Imaeda, Toshihiro [1 ]
Yokota, Akihiro [1 ]
Sogabe, Satoshi [1 ]
Kunugi, Akiyoshi [1 ]
Kuno, Haruhiko [1 ]
Kosugi, Yohei [1 ]
Kori, Masakuni [1 ]
Miki, Takashi [1 ]
Kimura, Haruhide [1 ]
Kuroita, Takanobu [1 ]
Kaku, Tomohiro [1 ]
机构
[1] Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
关键词
D O I
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
314
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页数:1
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