Discovery of TAK-137 and TAK-653, clinical candidates of α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid receptor potentiators with reduced agonistic activities
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作者:
Nakamura, Shinji
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Nakamura, Shinji
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Toyofuku, Masashi
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Toyofuku, Masashi
[1
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Honda, Eiji
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Honda, Eiji
[1
]
Imaeda, Toshihiro
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Imaeda, Toshihiro
[1
]
Yokota, Akihiro
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Yokota, Akihiro
[1
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Sogabe, Satoshi
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Sogabe, Satoshi
[1
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Kunugi, Akiyoshi
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kunugi, Akiyoshi
[1
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Kuno, Haruhiko
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kuno, Haruhiko
[1
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Kosugi, Yohei
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kosugi, Yohei
[1
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Kori, Masakuni
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kori, Masakuni
[1
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Miki, Takashi
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Miki, Takashi
[1
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Kimura, Haruhide
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kimura, Haruhide
[1
]
Kuroita, Takanobu
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kuroita, Takanobu
[1
]
Kaku, Tomohiro
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Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, JapanTakeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
Kaku, Tomohiro
[1
]
机构:
[1] Takeda Pharmaceut Co Ltd, Fujisawa, Kanagawa, Japan
机构:
Taisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, JapanTaisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, Japan
Koike, Hiroyuki
Iijima, Michihiko
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Taisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, JapanTaisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, Japan
Iijima, Michihiko
Kurosu, Shinsuke
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机构:
Taisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, JapanTaisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, Japan
Kurosu, Shinsuke
Chaki, Shigeyuki
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机构:
Taisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, JapanTaisho Pharmaceut Co Ltd, Mol Funct Pharmacol Labs, Discov Pharmacol, Kita Ku, Saitama 3319530, Japan
机构:
Ohio State Univ, Dept Neurol, Div Neuroimmunol, Columbus, OH 43210 USAOhio State Univ, Dept Neurol, Div Neuroimmunol, Columbus, OH 43210 USA
Pitt, David
Gonzales, Ernesto
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机构:
Washington Univ, Sch Med, Dept Neurol, St Louis, MO 63110 USA
Washington Univ, Sch Med, Hope Ctr Neurol Disorders, St Louis, MO 63110 USAOhio State Univ, Dept Neurol, Div Neuroimmunol, Columbus, OH 43210 USA
Gonzales, Ernesto
Cross, Anne H.
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机构:
Washington Univ, Sch Med, Dept Neurol, St Louis, MO 63110 USA
Washington Univ, Sch Med, Hope Ctr Neurol Disorders, St Louis, MO 63110 USAOhio State Univ, Dept Neurol, Div Neuroimmunol, Columbus, OH 43210 USA
Cross, Anne H.
Goldberg, Mark P.
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Washington Univ, Sch Med, Dept Neurol, St Louis, MO 63110 USA
Washington Univ, Sch Med, Hope Ctr Neurol Disorders, St Louis, MO 63110 USAOhio State Univ, Dept Neurol, Div Neuroimmunol, Columbus, OH 43210 USA